SCHEMBL3746150

SCHEMBL3746150

Cc1ccccc1-c1nc(-c2ccc3occc3c2)no1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 12/20 0.56
SMN1; SMN2 Q16637 10/20 0.56
RAB9A P51151 10/20 0.56
KDM4E B2RXH2 4/20 0.56
HPGD P15428 3/20 0.56
TSHR P16473 1/20 0.56
AHR P35869 1/20 0.56
S1PR1 P21453 2/20 0.54
MAPT P10636 5/20 0.49
TP53 P04637 3/20 0.49
RXFP1 Q9HBX9 1/20 0.49
MEN1 O00255 3/20 0.49
KMT2A Q03164 3/20 0.49
HSD17B10 Q99714 3/20 0.49
PKM P14618 2/20 0.49
GAA P10253 2/20 0.49
NFKB1 P19838 2/20 0.49
NFKB2 Q00653 2/20 0.49
RELA Q04206 2/20 0.49
L3MBTL1 Q9Y468 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3746152 0.90 NPC1 (0.59) NPC1SMN1; SMN2RAB9AS1PR1MAPT
SCHEMBL3743148 0.80 SMN1; SMN2 (0.68) NPC1SMN1; SMN2RAB9AKDM4EHPGD
SCHEMBL13417178 0.78 S1PR1 (0.62) NPC1SMN1; SMN2RAB9AKDM4ETSHR
SCHEMBL3747069 0.77 NPC1 (0.60) NPC1SMN1; SMN2RAB9AKDM4EHPGD
Dimethylamine SCHEMBL7961743 0.76 SMN1; SMN2 (0.67) NPC1SMN1; SMN2RAB9AKDM4EHPGD
SCHEMBL58788 0.74 NR1H4 (0.81) NPC1SMN1; SMN2RAB9AKDM4EHPGD
SCHEMBL28889002 0.73 S1PR1 (0.58) NPC1SMN1; SMN2RAB9AKDM4EHPGD
SCHEMBL23524328 0.73 NPC1 (0.49) NPC1SMN1; SMN2RAB9AKDM4EHPGD
SCHEMBL30355372 0.73 NPC1 (0.49) NPC1SMN1; SMN2RAB9AKDM4EHPGD
SCHEMBL13524984 0.72 S1PR1 (0.62) NPC1SMN1; SMN2RAB9AKDM4ES1PR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7834039-B2 Oxadiazole compounds ABBOTT LABORATORIES (US) 2010-11-16 US disclosed
US-7834039-B2 Oxadiazole compounds ABBOTT LABORATORIES (US) 2010-11-16 US disclosed
US-7834039-B2 Oxadiazole compounds ABBOTT LABORATORIES (US) 2010-11-16 US disclosed
EP-2109364-A1 NOVEL OXADIAZOLE COMPOUNDS Abbott Laboratories (US) 2009-10-21 EP disclosed
US-20080280876-A1 Novel oxadiazole compounds ABBVIE INC. 2008-11-13 US disclosed
US-20080280876-A1 Novel oxadiazole compounds ABBVIE INC. 2008-11-13 US disclosed
US-20080280876-A1 Novel oxadiazole compounds ABBVIE INC. 2008-11-13 US disclosed
WO-2008076356-A1 NOVEL OXADIAZOLE COMPOUNDS ABBOTT LABORATORIES (US) 2008-06-26 WO disclosed
WO-2008076356-A1 NOVEL OXADIAZOLE COMPOUNDS ABBOTT LABORATORIES (US) 2008-06-26 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080280876-A1 Novel oxadiazole compounds S1PR3, S1PR1, S1PR2 NPC1 1268/4885SMN1; SMN2 3564/4885RAB9A 2582/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.