Leucine

Leucine

SCHEMBL375261

CC(C)C(N)C(=O)O.CC(C)CC(N)C(=O)O.CC(C)[C@H](N)C(=O)O

nearest known ligand 0.78

Full drug profile on Sugi Atlas →

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SLC7A5 Q01650 2/20 0.78
SLC1A3 P43003 6/20 0.61
SLC1A2 P43004 6/20 0.61
SLC1A1 P43005 6/20 0.57
GRIK1 P39086 8/20 0.44
GRIK2 Q13002 5/20 0.44
GRM1 Q13255 1/20 0.43
GRM2 Q14416 1/20 0.43
RNPEP Q9H4A4 1/20 0.41
GRIA2 P42262 2/20 0.41
GRIA4 P48058 2/20 0.41
GRIK3 Q13003 2/20 0.41
GRIK5 Q16478 2/20 0.41
GRIA1 P42261 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Leucine SCHEMBL17184327 1.00 SLC7A5 (0.78) SLC7A5SLC1A3SLC1A2SLC1A1GRIK1
Leucine SCHEMBL4394463 1.00 SLC7A5 (0.78) SLC7A5SLC1A3SLC1A2SLC1A1GRIK1
Leucine SCHEMBL4401591 1.00 SLC7A5 (0.78) SLC7A5SLC1A3SLC1A2SLC1A1GRIK1
Leucine SCHEMBL466382 1.00 SLC7A5 (0.78) SLC7A5SLC1A3SLC1A2SLC1A1GRIK1
Leucine SCHEMBL28161805 1.00 SLC7A5 (0.78) SLC7A5SLC1A3SLC1A2SLC1A1GRIK1
Leucine SCHEMBL17184328 1.00 SLC7A5 (0.78) SLC7A5SLC1A3SLC1A2SLC1A1GRIK1
D-Leucine SCHEMBL11768667 1.00 SLC7A5 (0.78) SLC7A5SLC1A3SLC1A2SLC1A1GRIK1
Leucine SCHEMBL11305893 1.00 SLC7A5 (0.78) SLC7A5SLC1A3SLC1A2SLC1A1GRIK1
Leucine SCHEMBL466383 1.00 SLC7A5 (0.78) SLC7A5SLC1A3SLC1A2SLC1A1GRIK1
Leucine SCHEMBL2553000 0.96 SLC7A5 (0.72) SLC7A5SLC1A3SLC1A2SLC1A1GRIK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2408462-A1 Targeted delivery of chemotherapeutic agents Sanford-Burnham Medical Research Institute (US) 2012-01-25 EP disclosed
WO-2010108122-A1 TARGETED DELIVERY OF CHEMOTHERAPEUTIC AGENTS SANFORD-BURNHAM MEDICAL RESEARCH INSTITUTE (US) 2010-09-23 WO disclosed