SCHEMBL3754368

SCHEMBL3754368

Cc1c(COS(C)(=O)=O)nn(-c2ccc(Cl)cc2Cl)c1-c1ccc(Cl)s1

nearest known ligand 0.52

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 11/20 0.52
CNR2 P34972 11/20 0.52
OPRL1 P41146 6/20 0.43
KCNH2 Q12809 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3740310 0.82 CNR1 (0.55) CNR1CNR2OPRL1KCNH2
SCHEMBL3742041 0.82 CNR1 (0.57) CNR1CNR2OPRL1KCNH2
SCHEMBL1984928 0.75 CNR1 (0.65) CNR1CNR2
SCHEMBL4513948 0.75 CNR2 (0.70) CNR1CNR2
SCHEMBL1985291 0.75 CNR2 (0.70) CNR1CNR2
SCHEMBL1985913 0.74 CNR2 (0.59) CNR1CNR2
SCHEMBL3743339 0.74 OPRL1 (0.38) CNR1CNR2OPRL1KCNH2
SCHEMBL1983956 0.73 CNR2 (0.55) CNR1CNR2
SCHEMBL3747625 0.73 CNR1 (0.60) CNR1CNR2OPRL1KCNH2
SCHEMBL3742640 0.73 CNR1 (0.57) CNR1CNR2OPRL1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2068870-B1 THIOPHENE COMPOUNDS NAT HEALTH RESEARCH INSTITUTES (TW) 2013-03-27 EP disclosed
CN-101535260-B Thiophene compounds NAT HEALTH RESEARCH INSTITUTES 2012-07-04 CN disclosed
US-7834046-B2 Thiophene compounds NATIONAL HEALTH RESEARCH INSTITUTES (TW) 2010-11-16 US disclosed
CN-101535260-A Thiophene compounds NAT HEALTH RESEARCH INSTITUTES (CN) 2009-09-16 CN disclosed
EP-2068870-A2 THIOPHENE COMPOUNDS National Health Research Institutes (TW) 2009-06-17 EP disclosed
US-20090029969-A2 Thiophene Compounds NATIONAL HEALTH RESEARCH INSTITUTES (TW) 2009-01-29 US disclosed
WO-2008057681-A2 THIOPHENE COMPOUNDS NATIONAL HEALTH RESEARCH INSTITUTES (TW) 2008-05-15 WO disclosed
US-20080090810-A1 THIOPHENE COMPOUNDS NATIONAL HEALTH RESEARCH INSTITUTES (TW) 2008-04-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080090810-A1 THIOPHENE COMPOUNDS CNR1, CNR2, HTR2C CNR1 1/4885CNR2 2/4885OPRL1 4/4885
US-20090029969-A2 Thiophene Compounds CNR1, CNR2, HTR2C CNR1 1/4885CNR2 2/4885OPRL1 4/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.