SCHEMBL3765024

SCHEMBL3765024

CC1(C)CC(=O)c2sc(N3CCOCC3)c(-c3ccccc3Oc3ccccc3)c2C1

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 6/20 0.49
PIK3CA P42336 4/20 0.40
PIK3CD O00329 3/20 0.40
PIK3CG P48736 3/20 0.40
PIK3CB P42338 2/20 0.40
STK10 O94804 1/20 0.35
SLK Q9H2G2 1/20 0.35
POLB P06746 1/20 0.34
ALDH1A1 P00352 1/20 0.34
MAPT P10636 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
TDP2 O95551 1/20 0.34
HSD17B10 Q99714 1/20 0.34
PRKDC P78527 1/20 0.34
BUB1 O43683 2/20 0.33
CNR2 P34972 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3759992 0.89 BRD4 (0.47) BRD4PIK3CAPIK3CDPIK3CGPIK3CB
SCHEMBL3759255 0.86 BRD4 (0.52) BRD4PIK3CAPIK3CDPIK3CGPIK3CB
SCHEMBL3760389 0.82 BRD4 (0.46) BRD4PIK3CAPIK3CDPIK3CGPIK3CB
SCHEMBL3763827 0.81 PIK3CD (0.40) BRD4PIK3CAPIK3CDPIK3CGPIK3CB
SCHEMBL3766018 0.79 PRKDC (0.49) BRD4PIK3CAPIK3CDPIK3CGPIK3CB
SCHEMBL3758948 0.79 PIK3CD (0.42) BRD4PIK3CAPIK3CDPIK3CGPIK3CB
SCHEMBL3754814 0.78 PRKDC (0.46) BRD4PIK3CAPIK3CDPIK3CGPIK3CB
SCHEMBL3759838 0.78 PRKDC (0.48) BRD4PIK3CAPIK3CDPIK3CGPIK3CB
SCHEMBL3760606 0.78 PRKDC (0.46) BRD4PIK3CAPIK3CDPIK3CGPIK3CB
SCHEMBL3760440 0.77 PRKDC (0.51) BRD4PIK3CAPIK3CDPIK3CGPIK3CB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2029570-B1 FUSED THIOPHENE DERIVATIVES AS KINASE INHIBITORS UCB PHARMA SA (BE) 2014-10-15 EP disclosed
US-8324204-B2 Fused thiophene derivatives as kinase inhibitors UCB PHARMA SA (BE) 2012-12-04 US disclosed
US-20100305066-A1 Fused Thiophene Derivatives as Kinase Inhibitors UCB PHARMA S.A. (BE) 2010-12-02 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100305066-A1 Fused Thiophene Derivatives as Kinase Inhibitors PIKFYVE, PI4KA, PIK3CA BRD4 1041/4885PIK3CA 3/4885PIK3CD 9/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.