SCHEMBL37721

SCHEMBL37721

Fc1cccc(CC[Mg]Br)c1

nearest known ligand 0.57

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 3/20 0.57
SLC6A3 Q01959 2/20 0.47
IDO1 P14902 2/20 0.46
AGXT P21549 2/20 0.46
DRD2 P14416 1/20 0.45
SLC6A4 P31645 1/20 0.45
DAO P14920 2/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
MIF P14174 1/20 0.42
MAOB P27338 1/20 0.41
ALDH1A1 P00352 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11144848 0.89 TAAR1 (0.53) TAAR1SLC6A3IDO1AGXTDRD2
SCHEMBL3371633 0.80 TAAR1 (0.74) TAAR1SLC6A3IDO1AGXTDRD2
SCHEMBL1538033 0.79 TAAR1 (0.50) TAAR1SLC6A3IDO1AGXTDRD2
SCHEMBL11152261 0.78 TAAR1 (0.59) TAAR1IDO1AGXTMAOBSMN1; SMN2
SCHEMBL17552669 0.77 TAAR1 (0.63) TAAR1SLC6A3IDO1AGXTDRD2
SCHEMBL931383 0.77 TAAR1 (0.63) TAAR1SLC6A3IDO1AGXTDRD2
SCHEMBL30186558 0.77 TAAR1 (0.63) TAAR1SLC6A3IDO1AGXTDRD2
SCHEMBL11151686 0.76 TP53 (0.39) TAAR1IDO1MEN1KMT2AALDH1A1
SCHEMBL11152109 0.76 TAAR1 (0.57) TAAR1IDO1AGXTDAO
SCHEMBL11151588 0.76 TAAR1 (0.57) TAAR1IDO1DAOMAOBALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8796470-B2 Substituted octahydrocyclopenta[c]pyrroles as calcium channel modulators ABBVIE INC. (US) 2014-08-05 US disclosed
WO-2011149993-A2 SUBSTITUTED OCTAHYDROCYCLOPENTA[c]PYRROLES AS CALCIUM CHANNEL MODULATORS ABBOTT LABORATORIES (US) 2011-12-01 WO disclosed
US-20110294854-A1 SUBSTITUTED OCTAHYDROCYCLOPENTA[c]PYRROLES AS CALCIUM CHANNEL MODULATORS ABBOTT LABORATORIES (US) 2011-12-01 US disclosed
EP-0024943-B1 5,6,7-TRINOR-4,8-INTER-M-PHENYLENE PGI2 DERIVATIVES AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM TORAY INDUSTRIES, INC. (JP) 1983-08-17 EP disclosed
US-4301164-A FOR USE AS ANTIULCER AGENTS, HYPOTENSIVE AGENTS, ANTITHROMBOSIC AGENTS TORAY INDUSTRIES, INC. (JP) 1981-11-17 US disclosed
EP-0024943-A1 5,6,7-Trinor-4,8-inter-m-phenylene PGI2 derivatives and pharmaceutical compositions containing them TORAY INDUSTRIES, INC. (JP) 1981-03-11 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110294854-A1 SUBSTITUTED OCTAHYDROCYCLOPENTA[c]PYRROLES AS CALCIUM CHANNEL MODULATORS ORAI1, CACNA1E, RYR1 TAAR1 1163/4885SLC6A3 905/4885IDO1 2175/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.