SCHEMBL3772950

SCHEMBL3772950

O[C@@H]1CN(C2CCC(c3ccccc3)CC2)CCc2cc(OCc3ccccc3)ccc21

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 12/20 1.00
GRIN2B Q13224 12/20 1.00
HRH3 Q9Y5N1 4/20 0.62
CYP2D6 P10635 2/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3390701 1.00 GRIN1 (1.00) GRIN1GRIN2BHRH3CYP2D6
SCHEMBL3390698 1.00 GRIN1 (1.00) GRIN1GRIN2BHRH3CYP2D6
SCHEMBL3395790 1.00 GRIN1 (1.00) GRIN1GRIN2BHRH3CYP2D6
SCHEMBL18587456 0.85 GRIN2B (0.74) GRIN1GRIN2B
SCHEMBL3396820 0.85 GRIN2B (0.74) GRIN1GRIN2B
SCHEMBL3394780 0.85 GRIN2B (0.74) GRIN1GRIN2B
SCHEMBL3394777 0.85 GRIN2B (0.74) GRIN1GRIN2B
SCHEMBL3392243 0.82 GRIN1 (1.00) GRIN1GRIN2B
SCHEMBL3394459 0.82 GRIN1 (1.00) GRIN1GRIN2B
SCHEMBL3392245 0.82 GRIN1 (1.00) GRIN1GRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010122134-A1 NR2B-SELECTIVE NMDA-RECEPTOR ANTAGONISTS Westfälische Wilhelms Universität Münster (DE) 2010-10-28 WO disclosed