SCHEMBL37731

SCHEMBL37731

CC(=O)NC1(C)CCC2CN(Cc3ccccc3)CC21

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 4/20 0.42
CYP2D6 P10635 1/20 0.41
S1PR1 P21453 1/20 0.41
S1PR5 Q9H228 1/20 0.41
KMT2A Q03164 2/20 0.41
KDM4E B2RXH2 1/20 0.41
MEN1 O00255 1/20 0.41
ALDH1A1 P00352 1/20 0.41
RAB9A P51151 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
FUCA1 P04066 2/20 0.40
OPRM1 P35372 1/20 0.39
OPRD1 P41143 1/20 0.39
OPRK1 P41145 1/20 0.39
OPRL1 P41146 1/20 0.39
DRD2 P14416 1/20 0.39
DRD4 P21917 1/20 0.39
DRD3 P35462 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL38609 1.00 GRIN2B (0.42) GRIN2BCYP2D6S1PR1S1PR5KMT2A
SCHEMBL15908954 1.00 GRIN2B (0.42) GRIN2BCYP2D6S1PR1S1PR5KMT2A
SCHEMBL15908943 0.88 DRD4 (0.44) GRIN2BCYP2D6KMT2AMEN1DRD2
SCHEMBL37325 0.88 DRD4 (0.44) GRIN2BCYP2D6KMT2AMEN1DRD2
SCHEMBL37324 0.88 DRD4 (0.44) GRIN2BCYP2D6KMT2AMEN1DRD2
SCHEMBL15908932 0.81 KMT2A (0.48) GRIN2BCYP2D6KMT2AMEN1ALDH1A1
SCHEMBL15909047 0.81 KMT2A (0.48) GRIN2BCYP2D6KMT2AMEN1ALDH1A1
SCHEMBL37562 0.81 KMT2A (0.48) GRIN2BCYP2D6KMT2AMEN1ALDH1A1
SCHEMBL21737963 0.76 KMT2A (0.50) CYP2D6S1PR1S1PR5KMT2AKDM4E
SCHEMBL21797227 0.76 KMT2A (0.50) CYP2D6S1PR1S1PR5KMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011149993-A2 SUBSTITUTED OCTAHYDROCYCLOPENTA[c]PYRROLES AS CALCIUM CHANNEL MODULATORS ABBOTT LABORATORIES (US) 2011-12-01 WO claimed
WO-2011149993-A2 SUBSTITUTED OCTAHYDROCYCLOPENTA[c]PYRROLES AS CALCIUM CHANNEL MODULATORS ABBOTT LABORATORIES (US) 2011-12-01 WO disclosed