SCHEMBL377432

SCHEMBL377432

CC1CN(Cc2ccc(N(C)C(=O)N3CCC(Nc4ccccc4F)CC3)cc2)CCN1

nearest known ligand 0.56

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
MLNR O43193 20/20 0.56
CYP3A4 P08684 4/20 0.55
CYP2D6 P10635 1/20 0.54
KCNH2 Q12809 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL377786 1.00 MLNR (0.56) MLNRCYP3A4CYP2D6KCNH2
SCHEMBL377479 0.88 MLNR (0.49) MLNRCYP3A4CYP2D6KCNH2
SCHEMBL377805 0.87 MLNR (0.56) MLNRCYP3A4CYP2D6KCNH2
SCHEMBL377711 0.86 MLNR (0.74) MLNRCYP3A4CYP2D6KCNH2
SCHEMBL1704459 0.86 MLNR (0.74) MLNRCYP3A4CYP2D6KCNH2
SCHEMBL377798 0.85 KDM4E (0.49) MLNRCYP3A4
SCHEMBL377443 0.85 MLNR (0.76) MLNRCYP3A4CYP2D6KCNH2
SCHEMBL377832 0.85 MLNR (0.76) MLNRCYP3A4CYP2D6KCNH2
SCHEMBL377476 0.82 MLNR (0.64) MLNRCYP3A4CYP2D6KCNH2
SCHEMBL377498 0.82 MLNR (0.64) MLNRCYP3A4CYP2D6KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2029538-B1 BENZYLPIPERAZINE DERIVATIVES AS MOTILIN RECEPTOR ANTAGONISTS GLAXO GROUP LTD (GB) 2012-01-25 EP claimed