SCHEMBL3775862

SCHEMBL3775862

O=C(C[N+]12CCC(CC1)C(OC(=O)C(Cc1ccccc1)Nc1ccccc1)C2)c1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CHRM3 P20309 18/20 0.42
CHRM2 P08172 16/20 0.42
CHRM1 P11229 9/20 0.41
NPSR1 Q6W5P4 1/20 0.40
CYP2D6 P10635 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13282721 1.00 CHRM3 (0.42) CHRM3CHRM2CHRM1NPSR1CYP2D6
SCHEMBL3782039 1.00 CHRM3 (0.42) CHRM3CHRM2CHRM1NPSR1CYP2D6
SCHEMBL3775856 1.00 CHRM3 (0.42) CHRM3CHRM2CHRM1NPSR1CYP2D6
Bromide SCHEMBL2542613 0.99 CHRM3 (0.44) CHRM3CHRM2CHRM1NPSR1
Bromide SCHEMBL2482100 0.99 CHRM3 (0.44) CHRM3CHRM2CHRM1NPSR1
Trifluoroacetic Acid SCHEMBL2482985 0.93 CHRM3 (0.41) CHRM3CHRM2CHRM1NPSR1
SCHEMBL3785004 0.88 CHRM3 (0.47) CHRM3CHRM2CHRM1
SCHEMBL13285508 0.88 CHRM3 (0.47) CHRM3CHRM2CHRM1
SCHEMBL3780154 0.88 CHRM3 (0.47) CHRM3CHRM2CHRM1
SCHEMBL3780152 0.88 CHRM3 (0.47) CHRM3CHRM2CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2376489-B1 ALKALOID AMINOESTER DERIVATIVES AND MEDICINAL COMPOSITION THEREOF CHIESI FARMA SPA (IT) 2015-04-22 EP claimed
US-8835682-B2 Alkaloid aminoester derivatives and medicinal composition thereof CHIESI FARMACEUTICI S.P.A. (IT) 2014-09-16 US disclosed
EP-2206712-A1 \"Alkaloid aminoester derivatives and medicinal composition thereof\ CHIESI FARMACEUTICI S.p.A. (IT) 2010-07-14 EP disclosed