SCHEMBL3782345

SCHEMBL3782345

CN(C)C(=O)c1ccc2c(c1)CCCO2

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTNNB1 P35222 7/20 0.57
WNT3A P56704 7/20 0.57
PRKCI P41743 1/20 0.50
TAS1R3 Q7RTX0 2/20 0.44
TAS1R1 Q7RTX1 2/20 0.44
ALDH1A1 P00352 1/20 0.43
GAA P10253 1/20 0.43
HPGD P15428 1/20 0.43
TSHR P16473 1/20 0.43
PIR O00625 1/20 0.43
HSF1 Q00613 1/20 0.43
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
PDK1 Q15118 1/20 0.42
PDK2 Q15119 1/20 0.42
PDK3 Q15120 1/20 0.42
PDK4 Q16654 1/20 0.42
CLK1 P49759 1/20 0.42
DYRK1A Q13627 1/20 0.42
DYRK1B Q9Y463 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19864447 0.91 PRKCI (0.57) CTNNB1WNT3APRKCITAS1R3TAS1R1
SCHEMBL1726294 0.83 CTNNB1 (0.61) CTNNB1WNT3APRKCITAS1R3TAS1R1
SCHEMBL875455 0.81 CTNNB1 (0.67) CTNNB1WNT3APRKCITAS1R3TAS1R1
SCHEMBL31262479 0.81 CTNNB1 (0.67) CTNNB1WNT3APRKCITAS1R3TAS1R1
SCHEMBL29654041 0.80 PRKCI (0.63) CTNNB1WNT3APRKCITAS1R3TAS1R1
SCHEMBL8319676 0.80 PRKCI (0.63) CTNNB1WNT3APRKCITAS1R3TAS1R1
SCHEMBL15969319 0.79 CTNNB1 (0.68) CTNNB1WNT3APRKCIALDH1A1HPGD
SCHEMBL28709593 0.79 TSHR (0.62) CTNNB1WNT3AALDH1A1GAAHPGD
SCHEMBL27312616 0.79 CTNNB1 (0.57) CTNNB1WNT3APRKCITAS1R3TAS1R1
SCHEMBL671055 0.79 CTNNB1 (0.57) CTNNB1WNT3APRKCITAS1R3TAS1R1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2234486-A1 BENZIMIDAZOLES AND ANALOGS AS RHO KINASE INHIBITORS The Scripps Research Institute (US) 2010-10-06 EP disclosed
WO-2009079011-A1 BENZIMIDAZOLES AND ANALOGS AS RHO KINASE INHIBITORS THE SCRIPPS RESEARCH INSTITUTE (US) 2009-06-25 WO disclosed