SCHEMBL378338

SCHEMBL378338

Cc1ccc2c(-c3nnc(SCCCN4C[C@@H]5C[C@@]5(c5ccc(C(F)(F)F)cc5)C4)n3C)ccc(F)c2n1

nearest known ligand 0.77

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 20/20 0.77
DRD3 P35462 19/20 0.77
DRD2 P14416 15/20 0.77
CYP1A2 P05177 1/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL378370 1.00 KCNH2 (0.77) KCNH2DRD3DRD2CYP1A2
SCHEMBL378337 1.00 KCNH2 (0.77) KCNH2DRD3DRD2CYP1A2
Hydrochloric Acid SCHEMBL4436139 0.99 KCNH2 (0.76) KCNH2DRD3DRD2CYP1A2
Hydrochloric Acid SCHEMBL4563583 0.99 KCNH2 (0.76) KCNH2DRD3DRD2CYP1A2
SCHEMBL378656 0.87 KCNH2 (1.00) KCNH2DRD3DRD2
Hydrochloric Acid SCHEMBL378536 0.87 KCNH2 (0.98) KCNH2DRD3DRD2
SCHEMBL378352 0.82 DRD3 (1.00) KCNH2DRD3DRD2CYP1A2
SCHEMBL378509 0.81 DRD3 (1.00) KCNH2DRD3DRD2CYP1A2
Hydrochloric Acid SCHEMBL397107 0.81 DRD3 (0.98) KCNH2DRD3DRD2CYP1A2
SCHEMBL3364262 0.81 DRD3 (0.79) KCNH2DRD3DRD2CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2060570-B1 Azabicyclo[3.1.0] hexane derivatives useful as modulators of dopamine D3 receptors GLAXO GROUP LTD (GB) 2012-01-25 EP claimed