Terbinafine

Terbinafine

SCHEMBL37843

CN(CC=CC#CC(C)(C)C)Cc1cccc2ccccc12

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 4/20 1.00
LMNA P02545 4/20 1.00
SLC6A2 P23975 3/20 1.00
SIGMAR1 Q99720 3/20 1.00
SQLE Q14534 3/20 1.00
ADRA2A P08913 2/20 1.00
CYP1A2 P05177 2/20 0.62
CYP2C19 P33261 2/20 0.62
NR1I2 O75469 2/20 0.62
HTR2A P28223 2/20 0.62
SLC6A4 P31645 2/20 0.62
KCNH2 Q12809 2/20 0.62
HTT P42858 2/20 0.62
DRD2 P14416 1/20 0.62
ADRA2C P18825 1/20 0.62
CNR1 P21554 1/20 0.62
ADRA1A P35348 1/20 0.62
OPRK1 P41145 1/20 0.62
SLC6A3 Q01959 1/20 0.62
EBP Q15125 1/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Terbinafine SCHEMBL2028187 1.00 CYP2D6 (1.00) CYP2D6LMNASLC6A2SIGMAR1SQLE
Terbinafine SCHEMBL2042785 1.00 CYP2D6 (1.00) CYP2D6LMNASLC6A2SIGMAR1SQLE
Terbinafine SCHEMBL29353314 1.00 CYP2D6 (1.00) CYP2D6LMNASLC6A2SIGMAR1SQLE
Terbinafine SCHEMBL31374681 1.00 CYP2D6 (1.00) CYP2D6LMNASLC6A2SIGMAR1SQLE
Terbinafine SCHEMBL29627458 1.00 CYP2D6 (1.00) CYP2D6LMNASLC6A2SIGMAR1SQLE
Terbinafine SCHEMBL36794 1.00 CYP2D6 (1.00) CYP2D6LMNASLC6A2SIGMAR1SQLE
Terbinafine SCHEMBL5279646 1.00 CYP2D6 (1.00) CYP2D6LMNASLC6A2SIGMAR1SQLE
Terbinafine SCHEMBL36795 0.99 CYP2D6 (0.97) CYP2D6LMNASLC6A2SIGMAR1SQLE
Terbinafine SCHEMBL3597456 0.99 CYP2D6 (0.97) CYP2D6LMNASLC6A2SIGMAR1SQLE
Terbinafine SCHEMBL29871278 0.99 CYP2D6 (0.97) CYP2D6LMNASLC6A2SIGMAR1SQLE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 32823 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2026106917-A1 EDIBLE TRANSMUCOSAL DRUG DELIVERY METHOD USING AN INTERMEDIATE CAPSULE AS A TEMPORARY VESSEL BioPhysics Pharma, Inc. (US) 2026-05-21 WO claimed
CN-122031290-A Percutaneous permeation promoting system and preparation method and application thereof 北京工商大学 2026-05-15 CN claimed
US-20260124224-A1 USE OF COMBINED COMPOSITION IN PREPARING DRUG FOR RESISTING FUNGAL AND BACTERIAL INFECTIONS NATIONAL CENTER FOR NANOSCIENCE AND TECHNOLOGY (CN) 2026-05-07 US claimed
EP-4255391-B1 LUMINOL FOR USE IN THE TREATMENT OF SEQUELAE OF A SARS-COV-2 INFECTION METRIOPHARM AG (CH) 2026-05-06 EP claimed
EP-4731194-A1 MATERIALS AND METHODS FOR MITIGATING THE PRESENCE OF NITROSAMINES IN PACKAGING USING AN ACTIVE AGENT CSP Technologies, Inc. (US) 2026-04-29 EP claimed
US-12605345-B2 Transdermal drug delivery system BioPhysics Pharma, Inc. (US) 2026-04-21 US claimed
US-20260102363-A1 TREATMENT METHOD AND ANTIFUNGAL COMPOSITION MOBERG PHARMA AB (SE) 2026-04-16 US claimed
US-20260102333-A1 TOPICAL DELIVERY OF ANTIFUNGAL AGENTS FOR TREATING FUNGAL INFECTIONS LYOTROPIC DELIVERY SYSTEMS Ltd (IL) 2026-04-16 US claimed
US-20260102419-A1 USE OF COMPOUNDS IN THE TREATMENT OF FUNGAL INFECTIONS BASILEA PHARMACEUTICA INTERNATIONAL AG, ALLSCHWIL (CH) 2026-04-16 US claimed
EP-3175865-B1 FUNCTIONAL PARTICLES, PROCESS TO OBTAIN THEM, AND THEIR APPLICATIONS SMART INOVATION LDA (PT) 2026-04-15 EP claimed
US-5214046-A Synergistic mixtures, inhibitors of sterol biosynthesis HOFFMANN-LA ROCHE INC. (US) 1993-05-25 US claimed
EP-0503988-A1 Compositions to treat onychomycoses SANDOZ LTD. (CH) 1992-09-16 EP claimed
EP-0399858-B1 CLEANSING COMPOSITION CONTAINING IN PARTICULAR NAFTIFINE AND/OR TERBINAFINE L'OREAL (FR) 1992-07-08 EP claimed
EP-0478456-A1 Antifungal composition in dry aerosol form SANDOZ LTD (CH) 1992-04-01 EP claimed
EP-0310122-B1 ANTIFUNGAL COMPOSITION KAKEN PHARMACEUTICAL CO., LTD. (JP) 1991-07-24 EP claimed
EP-0399858-A1 Cleansing composition containing in particular naftifine and/or terbinafine L'OREAL (FR) 1990-11-28 EP claimed
US-4920112-A SYNERGISTIC 25-AZASTEROL COMPOUND AND SQUALENE EPOXIDASE INHIBITOR MERCK & CO., INC. (US) 1990-04-24 US claimed
US-4894375-A FUNGISTATS, KETOCONAZOLE MERCK & CO., INC. (US) 1990-01-16 US claimed
EP-0339708-A2 Fungicidal compositions and method MERCK & CO. INC. (US) 1989-11-02 EP claimed
EP-0310122-A1 Antifungal composition KAKEN PHARMACEUTICAL CO., LTD. (JP) 1989-04-05 EP claimed