SCHEMBL378439

SCHEMBL378439

Cc1ncccc1-c1nnc(SCCCN2C[C@H]3C[C@]3(c3ccc(C(F)(F)F)cc3F)C2)n1C

nearest known ligand 0.80

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 20/20 0.80
KCNH2 Q12809 19/20 0.80
DRD2 P14416 16/20 0.80
DRD4 P21917 1/20 0.77
CYP2C19 P33261 1/20 0.60
CHRM1 P11229 1/20 0.60
CHRM3 P20309 1/20 0.60
CYP1A2 P05177 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL378710 1.00 DRD3 (0.80) DRD3KCNH2DRD2DRD4CYP2C19
SCHEMBL378438 1.00 DRD3 (0.80) DRD3KCNH2DRD2DRD4CYP2C19
Hydrochloric Acid SCHEMBL4554725 0.99 DRD3 (0.79) DRD3KCNH2DRD2DRD4CYP2C19
Hydrochloric Acid SCHEMBL378272 0.99 DRD3 (0.79) DRD3KCNH2DRD2DRD4CYP2C19
SCHEMBL378509 0.89 DRD3 (1.00) DRD3KCNH2DRD2CYP2C19CHRM1
Hydrochloric Acid SCHEMBL393148 0.88 DRD3 (0.98) DRD3KCNH2DRD2CYP2C19CHRM1
Hydrochloric Acid SCHEMBL4411986 0.88 DRD3 (0.98) DRD3KCNH2DRD2CYP2C19CHRM1
Hydrochloric Acid SCHEMBL393147 0.88 DRD3 (0.98) DRD3KCNH2DRD2CYP2C19CHRM1
SCHEMBL378544 0.88 DRD3 (0.78) DRD3KCNH2DRD2DRD4CYP2C19
Hydrochloric Acid SCHEMBL378624 0.87 DRD3 (0.76) DRD3KCNH2DRD2DRD4CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2060570-B1 Azabicyclo[3.1.0] hexane derivatives useful as modulators of dopamine D3 receptors GLAXO GROUP LTD (GB) 2012-01-25 EP disclosed