SCHEMBL3789249

SCHEMBL3789249

COc1ccc(CN2CCc3ccc(Br)cc32)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 5/20 0.54
HDAC6 Q9UBN7 5/20 0.54
CYP1A2 P05177 1/20 0.52
CYP3A4 P08684 1/20 0.52
CYP2D6 P10635 1/20 0.52
NFKB1 P19838 1/20 0.52
HTR2A P28223 1/20 0.52
HTR2C P28335 1/20 0.52
HTR2B P41595 1/20 0.52
HIF1A Q16665 1/20 0.52
GAA P10253 2/20 0.49
ALDH1A1 P00352 1/20 0.49
ALOX15 P16050 1/20 0.49
TSHR P16473 1/20 0.49
LMNA P02545 1/20 0.44
PMP22 Q01453 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
GFER P55789 1/20 0.44
ABCB1 P08183 1/20 0.44
ABCC1 P33527 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3797439 0.92 HDAC1 (0.60) HDAC1HDAC6CYP1A2CYP3A4CYP2D6
SCHEMBL3793050 0.85 HTR2A (0.56) HDAC1HDAC6CYP1A2CYP3A4CYP2D6
SCHEMBL18586068 0.82 GAA (0.51) HDAC1HDAC6CYP1A2HTR2AHTR2C
SCHEMBL1556025 0.82 HDAC1 (0.60) HDAC1HDAC6TYMS
SCHEMBL16030871 0.81 CYP1A2 (0.55) HDAC1HDAC6CYP1A2CYP3A4CYP2D6
SCHEMBL3085320 0.80 GAA (0.70) NFKB1GAAALDH1A1ALOX15TSHR
SCHEMBL1431418 0.80 GAA (0.51) HDAC1HDAC6CYP1A2HTR2AHTR2C
SCHEMBL24317184 0.79 GAA (0.44) HDAC1HDAC6GAAALDH1A1LMNA
SCHEMBL23674994 0.78 HDAC1 (0.53) HDAC1HDAC6ALDH1A1
SCHEMBL30100741 0.78 HDAC1 (0.53) HDAC1HDAC6ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010128152-A1 FUSED HETEROCYCLIC C-GLYCOSIDES FOR THE TREATMENT OF DIABETES NOVARTIS AG (CH) 2010-11-11 WO disclosed