SCHEMBL378983

SCHEMBL378983

Cc1ccc2c(-c3nnc(SCCCN4CC5C[C@]5(c5ccc(O)cc5)C4)n3C)cccc2n1

nearest known ligand 0.88

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 20/20 0.88
DRD3 P35462 19/20 0.88
DRD2 P14416 16/20 0.88

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL394165 1.00 KCNH2 (0.88) KCNH2DRD3DRD2
SCHEMBL378317 1.00 KCNH2 (0.88) KCNH2DRD3DRD2
SCHEMBL378984 1.00 KCNH2 (0.88) KCNH2DRD3DRD2
SCHEMBL13079521 1.00 KCNH2 (0.88) KCNH2DRD3DRD2
SCHEMBL11911780 1.00 KCNH2 (0.88) KCNH2DRD3DRD2
Hydrochloric Acid SCHEMBL378459 0.99 KCNH2 (0.86) KCNH2DRD3DRD2
SCHEMBL5245524 0.94 KCNH2 (1.00) KCNH2DRD3DRD2
SCHEMBL5245984 0.94 KCNH2 (1.00) KCNH2DRD3DRD2
SCHEMBL378384 0.94 KCNH2 (1.00) KCNH2DRD3DRD2
SCHEMBL5245761 0.94 KCNH2 (1.00) KCNH2DRD3DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2060570-B1 Azabicyclo[3.1.0] hexane derivatives useful as modulators of dopamine D3 receptors GLAXO GROUP LTD (GB) 2012-01-25 EP claimed