SCHEMBL379029

SCHEMBL379029

N#Cc1cc(F)ccc1Oc1ccc2c(cnn2CCO)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP4K4 O95819 1/20 0.46
ABL1 P00519 1/20 0.46
NTRK1 P04629 1/20 0.46
FYN P06241 1/20 0.46
LYN P07948 1/20 0.46
RET P07949 1/20 0.46
BCR P11274 1/20 0.46
FGFR1 P11362 1/20 0.46
BRAF P15056 1/20 0.46
EPHA1 P21709 1/20 0.46
EPHA2 P29317 1/20 0.46
ABL2 P42684 1/20 0.46
FRK P42685 1/20 0.46
MAPK9 P45984 1/20 0.46
MAPKAPK2 P49137 1/20 0.46
IRAK1 P51617 1/20 0.46
MAPK10 P53779 1/20 0.46
EPHB3 P54753 1/20 0.46
EPHB4 P54760 1/20 0.46
CDK5 Q00535 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15995279 0.93 MAP4K4 (0.43) MAP4K4ABL1NTRK1FYNLYN
SCHEMBL12216031 0.89 AR (0.41) MAP4K4ABL1NTRK1FYNLYN
SCHEMBL2448337 0.87 MAPK14 (0.40) MAP4K4ABL1NTRK1FYNLYN
SCHEMBL12216030 0.85 MAP4K4 (0.40) MAP4K4ABL1NTRK1FYNLYN
SCHEMBL2446966 0.85 AR (0.41) MAP4K4ABL1NTRK1FYNLYN
SCHEMBL2444724 0.84 AR (0.40) ARSLC22A12CYP2C8CYP2C9CYP2C19
SCHEMBL2440738 0.84 HTR2A (0.50) MAPK14ARSLC22A12HTR2AHTR2C
SCHEMBL17407527 0.84 LYN (0.52) MAP4K4ABL1NTRK1FYNLYN
SCHEMBL15995520 0.84 MAP4K4 (0.54) MAP4K4ABL1NTRK1FYNLYN
SCHEMBL2445697 0.83 AR (0.44) ARSLC22A12CYP2C8CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 52 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4069792-A1 MICHAEL REACTION-CURING HYBRID SYSTEM FOR USE IN CHEMICAL FASTENING TECHNOLOGY fischerwerke GmbH & Co. KG (DE) 2022-10-12 EP claimed
WO-2021110621-A1 MICHAEL REACTION-CURING HYBRID SYSTEM FOR USE IN CHEMICAL FASTENING TECHNOLOGY FISCHERWERKE GMBH & CO. KG (DE) 2021-06-10 WO claimed
WO-2021110622-A1 MICHAEL REACTION-CURING SYNTHETIC RESIN FOR USE IN CHEMICAL FASTENING TECHNOLOGY FISCHERWERKE GMBH & CO. KG (DE) 2021-06-10 WO claimed
WO-2016173960-A1 OPTIMIZED SYNTHESIS OF PREGABALIN AND 4-AMINOBUTANE ACID USING AN IMPROVED METHOD FOR PRODUCING CONJUGATED NITROALKENES K.H.S. PHARMA HOLDING GMBH (DE) 2016-11-03 WO claimed
EP-3668721-B1 METHOD FOR PRODUCING A FILM-COATED ARTICLE AND FILM-COATED ARTICLE LEONHARD KURZ STIFTUNG & CO KG (DE) 2024-05-29 EP disclosed
WO-2024012829-A1 POLYMER COMPOSITION WHICH CAN BE CURED AT ROOM TEMPERATURE AND WHICH IS MADE OF POLYALDEHYDE AND POLYMALONATE SIKA TECHNOLOGY AG (CH) 2024-01-18 WO disclosed
WO-2024012826-A1 POLYMER HAVING ALDEHYDE GROUPS SIKA TECHNOLOGY AG (CH) 2024-01-18 WO disclosed
WO-2023186460-A1 FILM, FILM-COATED OBJECT AND METHOD FOR PRODUCING A FILM-COATED OBJECT LEONHARD KURZ STIFTUNG & CO. KG (DE) 2023-10-05 WO disclosed
EP-4069792-A1 MICHAEL REACTION-CURING HYBRID SYSTEM FOR USE IN CHEMICAL FASTENING TECHNOLOGY fischerwerke GmbH & Co. KG (DE) 2022-10-12 EP disclosed
WO-2021110621-A1 MICHAEL REACTION-CURING HYBRID SYSTEM FOR USE IN CHEMICAL FASTENING TECHNOLOGY FISCHERWERKE GMBH & CO. KG (DE) 2021-06-10 WO disclosed
WO-2021110622-A1 MICHAEL REACTION-CURING SYNTHETIC RESIN FOR USE IN CHEMICAL FASTENING TECHNOLOGY FISCHERWERKE GMBH & CO. KG (DE) 2021-06-10 WO disclosed
EP-3668721-A2 TRANSFER FILM, METHOD FOR PRODUCING A FILM-COATED ARTICLE AND FILM-COATED ARTICLE Leonhard Kurz Stiftung & Co. KG (DE) 2020-06-24 EP disclosed
EP-1981851-A1 KINASE INHIBITORS AND METHODS OF USE THEREOF Array Biopharma, Inc. (US) 2008-10-22 EP disclosed
EP-1648894-B1 METHOD FOR THE PRODUCTION OF OH PROTECTED [4-(2.6-DIAMINO-9H-PURINE-9-YL)- 1.3-DIOXOLANE-2-YL]METHANOL DERIVATIVES WACKER CHEMIE AG (DE) 2007-09-12 EP disclosed
WO-2007089646-A1 KINASE INHIBITORS AND METHODS OF USE THEREOF ARRAY BIOPHARMA INC. (US) 2007-08-09 WO disclosed
WO-2007089646-A1 KINASE INHIBITORS AND METHODS OF USE THEREOF ARRAY BIOPHARMA INC. (US) 2007-08-09 WO disclosed
EP-1648894-A1 METHOD FOR THE PRODUCTION OF OH PROTECTED [4-(2.6-DIAMINO-9H-PURINE-9-YL)- 1.3-DIOXOLANE-2-YL]METHANOL DERIVATIVES Wacker Chemie AG (DE) 2006-04-26 EP disclosed
WO-2005012302-A1 METHOD FOR THE PRODUCTION OF OH PROTECTED [4-(2.6-DIAMINO-9H-PURINE-9-YL)- 1.3-DIOXOLANE-2-YL]METHANOL DERIVATIVES WACKER CHEMIE AG (DE) 2005-02-10 WO disclosed
EP-0683154-B1 Diisocyanates, process for their preparation and their use BAYER AG (DE) 1998-08-19 EP disclosed
EP-0683154-A1 Diisocyanates, process for their preparation and their use BAYER AG (DE) 1995-11-22 EP disclosed