SCHEMBL3790448

SCHEMBL3790448

COC(=O)c1ccnc(-c2ccc(-c3ccc4[nH]ccc4c3)cc2)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK8 P49336 1/20 0.54
KDM4E B2RXH2 2/20 0.51
KDM4C Q9H3R0 2/20 0.51
KDM6B O15054 1/20 0.51
KDM5C P41229 1/20 0.51
KDM2A Q9Y2K7 1/20 0.51
KDM3A Q9Y4C1 1/20 0.51
PTGS2 P35354 1/20 0.46
JMJD6 Q6NYC1 1/20 0.46
HDAC2 Q92769 1/20 0.44
ALDH1A1 P00352 1/20 0.44
KDR P35968 1/20 0.44
NPC1 O15118 1/20 0.43
ABL1 P00519 2/20 0.43
CYP11B1 P15538 2/20 0.42
CYP11B2 P19099 2/20 0.42
CYP17A1 P05093 1/20 0.42
CHRNB4 P30926 1/20 0.42
CHRNA3 P32297 1/20 0.42
CHRNA7 P36544 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31464238 0.96 KDM4E (0.55) CDK8KDM4EKDM4CKDM6BKDM5C
SCHEMBL1646994 0.96 KDM4E (0.55) CDK8KDM4EKDM4CKDM6BKDM5C
SCHEMBL3788730 0.88 KDM4E (0.46) CDK8KDM4EKDM4CKDM6BKDM5C
SCHEMBL3789719 0.84 HDAC6 (0.54) PTGS2HDAC2NPC1ABL1CYP11B1
SCHEMBL1646106 0.83 JMJD6 (0.55) CDK8JMJD6KDR
SCHEMBL10819449 0.82 CDK8 (0.50) CDK8KDM4CPTGS2KDRNPC1
SCHEMBL20476711 0.81 KDM4E (0.58) CDK8KDM4EKDM4CKDM6BKDM5C
SCHEMBL1648927 0.79 CDK8 (0.45) CDK8KDM4EPTGS2HDAC2ALDH1A1
SCHEMBL27997808 0.79 KDM4E (0.69) KDM4EKDM4CKDM6BKDM5CKDM2A
SCHEMBL3718393 0.78 KDM4E (0.68) KDM4EKDM4CKDM6BKDM5CKDM2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010100475-A1 HYDROXAMIC ACID DERIVATIVES AS GRAM-NEGATIVE ANTIBACTERIAL AGENTS ASTRAZENECA AB (SE) 2010-09-10 WO disclosed
WO-2010100475-A1 HYDROXAMIC ACID DERIVATIVES AS GRAM-NEGATIVE ANTIBACTERIAL AGENTS ASTRAZENECA AB (SE) 2010-09-10 WO disclosed