SCHEMBL3790886

SCHEMBL3790886

NC(=O)OCCC(=O)N1CCC2(CC1)NC(=O)c1sc(-c3ccncc3)cc1N2

nearest known ligand 0.58

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ROCK1 Q13464 14/20 0.58
CDC7 O00311 13/20 0.58
DBF4 Q9UBU7 13/20 0.58
CCNE1 P24864 13/20 0.58
CDK2 P24941 13/20 0.58
ITGB3 P05106 4/20 0.33
ITGA2B P08514 4/20 0.33
NAMPT P43490 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32
TSHR P16473 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL613680 0.89 ROCK1 (0.60) ROCK1CDC7DBF4CCNE1CDK2
SCHEMBL613701 0.86 CDC7 (0.66) ROCK1CDC7DBF4CCNE1CDK2
SCHEMBL613816 0.85 ROCK1 (0.59) ROCK1CDC7DBF4CCNE1CDK2
SCHEMBL613656 0.84 ROCK1 (0.62) ROCK1CDC7DBF4CCNE1CDK2
SCHEMBL613682 0.83 ROCK1 (0.59) ROCK1CDC7DBF4CCNE1CDK2
SCHEMBL613280 0.83 CDC7 (0.70) ROCK1CDC7DBF4CCNE1CDK2
SCHEMBL612621 0.82 CDC7 (0.62) ROCK1CDC7DBF4CCNE1CDK2
SCHEMBL612136 0.81 ROCK1 (0.70) ROCK1CDC7DBF4CCNE1CDK2
SCHEMBL612014 0.81 ROCK1 (0.61) ROCK1CDC7DBF4CCNE1CDK2
SCHEMBL614242 0.81 ROCK1 (0.66) ROCK1CDC7DBF4CCNE1CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010101302-A1 THIENOPYRIMIDINE AS CDC7 KINASE INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-09-10 WO disclosed