SCHEMBL3792633

SCHEMBL3792633

Nc1cc(F)c(-c2ccnc(N)n2)c(F)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 3/20 0.47
AURKA O14965 2/20 0.47
PRKACA P17612 1/20 0.47
ADORA2A P29274 1/20 0.47
KMO O15229 1/20 0.45
FEN1 P39748 2/20 0.43
MAP3K14 Q99558 2/20 0.43
MAPK14 Q16539 1/20 0.43
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42
CDK5 Q00535 1/20 0.42
CDK5R1 Q15078 1/20 0.42
HSP90AB1 P08238 1/20 0.42
PTK2 Q05397 1/20 0.42
GRM4 Q14833 1/20 0.41
GSK3B P49841 1/20 0.41
CDK2 P24941 2/20 0.40
CDK4 P11802 1/20 0.40
CCNE1 P24864 1/20 0.40
CHUK O15111 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28513246 0.83 HSP90AA1 (0.53) HSP90AA1AURKAPRKACAADORA2AKMO
SCHEMBL30507455 0.83 HSP90AA1 (0.53) HSP90AA1AURKAPRKACAADORA2AKMO
SCHEMBL3792630 0.80 CDC7 (0.47) PRKACAMAPK14CDK5GSK3BCDK2
SCHEMBL18495643 0.75 FEN1 (0.48) HSP90AA1AURKAPRKACAADORA2AKMO
SCHEMBL3393995 0.73 HSP90AA1 (0.55) HSP90AA1AURKAPRKACAADORA2AKMO
SCHEMBL27159221 0.72 FEN1 (0.54) HSP90AA1AURKAPRKACAADORA2AKMO
SCHEMBL20467870 0.71 MAP3K14 (0.45) HSP90AA1AURKAPRKACAADORA2AKMO
SCHEMBL30353577 0.70 FEN1 (0.57) HSP90AA1AURKAPRKACAADORA2AFEN1
SCHEMBL5140478 0.70 FEN1 (0.57) HSP90AA1AURKAPRKACAADORA2AFEN1
SCHEMBL30775416 0.70 MAP3K14 (0.57) PRKACAKMOFEN1MAP3K14KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2234618-A1 BENZOPYRANS AND ANALOGS AS RHO KINASE INHIBITORS The Scripps Research Institute (US) 2010-10-06 EP disclosed
WO-2009079008-A1 BENZOPYRANS AND ANALOGS AS RHO KINASE INHIBITORS FENG YANGBO (US) 2009-06-25 WO disclosed