SCHEMBL3794590

SCHEMBL3794590

CN(C)C1CCN(c2ccc3nc(C(=O)c4ccnc(-c5ccc6c(c5)OCCO6)c4)[nH]c3c2)CC1.CN(C)C1CCN(c2ccc3nc(C(=O)c4ccnc(-c5cncc6ccccc56)c4)[nH]c3c2F)CC1

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 5/20 0.72
CCND1 P24385 5/20 0.72
CDK1 P06493 5/20 0.72
CCND3 P30281 4/20 0.72
CDK6 Q00534 4/20 0.72
CCNB1 P14635 3/20 0.72
CCNA2 P20248 3/20 0.72
CDK2 P24941 3/20 0.72
CCNA1 P78396 3/20 0.72
KDR P35968 3/20 0.34
RET P07949 2/20 0.34
PDCD1 Q15116 1/20 0.34
CD274 Q9NZQ7 1/20 0.34
MTOR P42345 3/20 0.33
PIK3CA P42336 1/20 0.33
ERBB2 P04626 1/20 0.33
BRD4 O60885 1/20 0.33
CREBBP Q92793 1/20 0.32
PDGFRB P09619 1/20 0.32
FGFR1 P11362 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL108773 0.87 CDK4 (0.73) CDK4CCND1CDK1CCND3CDK6
SCHEMBL112922 0.84 CDK4 (0.73) CDK4CCND1CDK1CCND3CDK6
SCHEMBL111812 0.80 CDK4 (0.89) CDK4CCND1CDK1CCND3CDK6
Hydrochloric Acid SCHEMBL175288 0.79 CDK4 (0.87) CDK4CCND1CDK1CCND3CDK6
SCHEMBL114340 0.78 CDK4 (0.84) CDK4CCND1CDK1CCND3CDK6
SCHEMBL2129207 0.76 CDK4 (0.78) CDK4CCND1CDK1CCND3CDK6
SCHEMBL110592 0.75 CDK4 (0.77) CDK4CCND1CDK1CCND3CDK6
SCHEMBL111954 0.75 CDK4 (1.00) CDK4CCND1CDK1CCND3CDK6
SCHEMBL109669 0.74 CDK4 (0.79) CDK4CCND1CDK1CCND3CDK6
SCHEMBL111810 0.74 CDK4 (0.83) CDK4CCND1CDK1CCND3CDK6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010125402-A1 IMIDAZOLE DERIVATIVES AND THEIR USE AS MODULATORS OF CYCLIN DEPENDENT KINASES NOVARTIS AG (CH) 2010-11-04 WO claimed