SCHEMBL3800622

SCHEMBL3800622

COC(=O)N[C@H](C(=O)N[C@@H](Cc1ccc(-c2ccccn2)cc1)C[C@H](O)[C@H](Cc1ccc(-c2ccccn2)cc1)NC(=O)[C@H](NC(=O)O)C(C)(C)C)C(C)(C)C

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 4/20 0.71
CTSD P07339 3/20 0.71
UGT1A1 P22309 3/20 0.69
ABCB11 O95342 2/20 0.69
ABCB1 P08183 2/20 0.69
ABCG2 Q9UNQ0 2/20 0.69
MLNR O43193 1/20 0.69
NR1I2 O75469 1/20 0.69
SLCO2B1 O94956 1/20 0.69
CCKAR P32238 1/20 0.69
OPRK1 P41145 1/20 0.69
GHSR Q92847 1/20 0.69
SLCO1B3 Q9NPD5 1/20 0.69
SLCO1B1 Q9Y6L6 1/20 0.69
KCNH2 Q12809 2/20 0.53
CA2 P00918 1/20 0.47
MME P08473 5/20 0.41
ABCC3 O15438 1/20 0.38
ABCC4 O15439 1/20 0.38
PGR P06401 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2436384 1.00 CYP3A4 (0.71) CYP3A4CTSDUGT1A1ABCB11ABCB1
SCHEMBL6428583 1.00 CYP3A4 (0.71) CYP3A4CTSDUGT1A1ABCB11ABCB1
SCHEMBL3803571 0.99 CYP3A4 (0.72) CYP3A4CTSDUGT1A1ABCB11ABCB1
SCHEMBL2435212 0.99 CYP3A4 (0.72) CYP3A4CTSDUGT1A1ABCB11ABCB1
SCHEMBL3804570 0.99 CYP3A4 (0.72) CYP3A4CTSDUGT1A1ABCB11ABCB1
SCHEMBL2435678 0.99 CYP3A4 (0.72) CYP3A4CTSDUGT1A1ABCB11ABCB1
SCHEMBL2433927 0.99 CYP3A4 (0.72) CYP3A4CTSDUGT1A1ABCB11ABCB1
SCHEMBL4250162 0.97 CYP3A4 (0.71) CYP3A4CTSDUGT1A1ABCB11ABCB1
SCHEMBL2436783 0.97 CYP3A4 (0.71) CYP3A4CTSDUGT1A1ABCB11ABCB1
SCHEMBL2436758 0.97 CYP3A4 (0.71) CYP3A4CTSDUGT1A1ABCB11ABCB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2266971-A2 Hiv protease inhibiting compounds Abbott Laboratories (US) 2010-12-29 EP disclosed