SCHEMBL3812290

SCHEMBL3812290

Nc1ccccc1NC(=O)c1cc2ccc(CCNCc3ccc(Cl)cc3)cc2s1

nearest known ligand 0.58

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 14/20 0.58
HDAC2 Q92769 4/20 0.56
DHPS P49366 1/20 0.45
PRSS12 P56730 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3575662 0.92 HDAC1 (0.60) HDAC1HDAC2DHPS
SCHEMBL3814883 0.90 HDAC1 (0.60) HDAC1HDAC2DHPS
SCHEMBL3810635 0.90 HDAC1 (0.58) HDAC1HDAC2
SCHEMBL3819259 0.88 HDAC1 (0.55) HDAC1HDAC2
SCHEMBL3820750 0.86 HDAC1 (0.63) HDAC1HDAC2DHPS
SCHEMBL3820287 0.85 HDAC1 (0.56) HDAC1HDAC2
SCHEMBL3565708 0.85 HDAC1 (0.71) HDAC1HDAC2
SCHEMBL5051806 0.84 HDAC1 (0.57) HDAC1HDAC2DHPS
SCHEMBL3570046 0.84 HDAC1 (0.60) HDAC1HDAC2DHPS
SCHEMBL3579612 0.83 HDAC2 (0.70) HDAC1HDAC2PRSS12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1874295-A4 BENZOTHIOPHENE DERIVATIVES MERCK & CO INC (US) 2009-08-12 EP disclosed
EP-1874295-A1 BENZOTHIOPHENE DERIVATIVES Merck & Co., Inc. (US) 2008-01-09 EP disclosed
WO-2006115845-A1 BENZOTHIOPHENE DERIVATIVES MERCK & CO., INC. (US) 2006-11-02 WO disclosed