SCHEMBL3818909

SCHEMBL3818909

COc1ccc(CN(C)CCc2ccc3cc(C(=O)Nc4ccccc4N)sc3c2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 13/20 0.47
HDAC2 Q92769 5/20 0.47
HDAC3 O15379 5/20 0.47
NCOR2 Q9Y618 3/20 0.47
HDAC10 Q969S8 2/20 0.47
HDAC4 P56524 1/20 0.46
HDAC7 Q8WUI4 1/20 0.46
HDAC11 Q96DB2 1/20 0.46
HDAC8 Q9BY41 1/20 0.46
HDAC6 Q9UBN7 1/20 0.46
HDAC9 Q9UKV0 1/20 0.46
HDAC5 Q9UQL6 1/20 0.46
ACKR3 P25106 2/20 0.44
NCOR1 O75376 1/20 0.44
MEN1 O00255 1/20 0.42
ALDH1A1 P00352 1/20 0.42
GAA P10253 1/20 0.42
KMT2A Q03164 1/20 0.42
CLK1 P49759 2/20 0.42
DYRK1A Q13627 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3811882 0.89 HDAC1 (0.47) HDAC1HDAC2HDAC3NCOR2HDAC10
SCHEMBL3814954 0.86 HDAC1 (0.46) HDAC1HDAC2HDAC3NCOR2HDAC10
SCHEMBL3571690 0.86 HDAC2 (0.48) HDAC1HDAC2HDAC3NCOR2HDAC10
SCHEMBL3563760 0.85 HDAC1 (0.51) HDAC1HDAC2HDAC3NCOR2HDAC10
SCHEMBL3819259 0.84 HDAC1 (0.55) HDAC1HDAC2HDAC3NCOR2HDAC10
SCHEMBL3579753 0.83 HDAC1 (0.57) HDAC1HDAC2HDAC3NCOR2HDAC10
SCHEMBL3810239 0.83 HDAC2 (0.57) HDAC1HDAC2HDAC3NCOR2HDAC10
SCHEMBL3563357 0.83 HDAC2 (0.46) HDAC1HDAC2HDAC3NCOR2HDAC10
SCHEMBL3820228 0.82 HDAC2 (0.52) HDAC1HDAC2HDAC3NCOR2HDAC10
SCHEMBL3810237 0.82 HDAC2 (0.51) HDAC1HDAC2HDAC3NCOR2HDAC10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1874295-A4 BENZOTHIOPHENE DERIVATIVES MERCK & CO INC (US) 2009-08-12 EP claimed
EP-1874295-A1 BENZOTHIOPHENE DERIVATIVES Merck & Co., Inc. (US) 2008-01-09 EP claimed
WO-2006115845-A1 BENZOTHIOPHENE DERIVATIVES MERCK & CO., INC. (US) 2006-11-02 WO claimed
EP-1874295-A4 BENZOTHIOPHENE DERIVATIVES MERCK & CO INC (US) 2009-08-12 EP disclosed
EP-1874295-A1 BENZOTHIOPHENE DERIVATIVES Merck & Co., Inc. (US) 2008-01-09 EP disclosed
WO-2006115845-A1 BENZOTHIOPHENE DERIVATIVES MERCK & CO., INC. (US) 2006-11-02 WO disclosed