SCHEMBL3826424

SCHEMBL3826424

Cc1ccc(NC(=O)c2cc(N3CCN(C)CC3)cc(C(F)(F)F)c2)cc1Nc1ncncc1-c1cc(NC2CC2)ncn1

nearest known ligand 0.63

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
BRAF P15056 14/20 0.63
LYN P07948 3/20 0.54
CSF1R P07333 2/20 0.54
RAF1 P04049 1/20 0.54
SRC P12931 3/20 0.53
INSR P06213 2/20 0.53
LCK P06239 2/20 0.53
KDR P35968 2/20 0.53
HCK P08631 1/20 0.53
ABL1 P00519 2/20 0.49
TEK Q02763 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3830584 0.93 BRAF (0.55) BRAFLYNCSF1RRAF1SRC
SCHEMBL3829713 0.93 BRAF (0.54) BRAFLYNRAF1SRCINSR
SCHEMBL3830996 0.91 BRAF (0.59) BRAFLYNCSF1RRAF1SRC
SCHEMBL3589285 0.90 BRAF (0.60) BRAFLYNCSF1RRAF1SRC
SCHEMBL3823342 0.87 LCK (0.65) BRAFLYNRAF1SRCINSR
SCHEMBL3823481 0.85 KDR (0.64) BRAFLYNCSF1RSRCINSR
SCHEMBL3822904 0.84 KDR (0.52) BRAFLYNCSF1RRAF1SRC
SCHEMBL3585148 0.83 BRAF (0.52) BRAFLYNCSF1RRAF1SRC
SCHEMBL3585600 0.82 LYN (0.57) BRAFLYNCSF1RRAF1SRC
SCHEMBL3586403 0.82 BRAF (0.61) BRAFLYNCSF1RRAF1SRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090069327-A1 COMPOUNDS AND COMPOSITIONS AS PROTEIN KINASE INHIBITORS IRM LLC (BM) 2009-03-12 US claimed
US-20090069327-A1 COMPOUNDS AND COMPOSITIONS AS PROTEIN KINASE INHIBITORS IRM LLC (BM) 2009-03-12 US disclosed
US-20090069327-A1 COMPOUNDS AND COMPOSITIONS AS PROTEIN KINASE INHIBITORS IRM LLC (BM) 2009-03-12 US disclosed
US-20090069327-A1 COMPOUNDS AND COMPOSITIONS AS PROTEIN KINASE INHIBITORS IRM LLC (BM) 2009-03-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090069327-A1 COMPOUNDS AND COMPOSITIONS AS PROTEIN KINASE INHIBITORS SRC, BMX, FYN BRAF 28/4885LYN 12/4885CSF1R 782/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.