SCHEMBL3828049

SCHEMBL3828049

CCCCc1ccc(-c2cnc3c(c2)c(O)c(C(=O)NCC(=O)O)c(=O)n3C)cc1

nearest known ligand 0.49

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
EGLN1 Q9GZT9 5/20 0.49
L3MBTL1 Q9Y468 1/20 0.44
HIF1A Q16665 12/20 0.44
EP300 Q09472 1/20 0.43
KAT2A Q92830 1/20 0.43
KAT2B Q92831 1/20 0.43
CNR2 P34972 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2576461 0.89 CNR2 (0.43) EGLN1L3MBTL1EP300KAT2AKAT2B
SCHEMBL2576312 0.89 EGLN1 (0.51) EGLN1L3MBTL1HIF1A
SCHEMBL2582204 0.86 EGLN1 (0.60) EGLN1HIF1A
SCHEMBL2581097 0.85 HIF1A (0.57) EGLN1HIF1A
SCHEMBL2585485 0.84 EGLN1 (0.51) EGLN1HIF1A
SCHEMBL2583340 0.83 EGLN1 (0.56) EGLN1HIF1A
SCHEMBL2578875 0.83 EGLN1 (0.52) EGLN1HIF1A
SCHEMBL2582349 0.82 EGLN1 (0.60) EGLN1HIF1A
SCHEMBL2574737 0.82 EGLN1 (0.52) EGLN1HIF1A
SCHEMBL2578353 0.81 HIF1A (0.51) EGLN1HIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2097416-A1 AZAQUINOLONE BASED COMPOUNDS EXHIBITING PROLYL HYDROXYLASE INHIBITORY ACTIVITY, COMPOSITIONS, AND USES THEREOF Amgen, Inc (US) 2009-09-09 EP disclosed
WO-2008076425-A1 AZAQUINOLONE BASED COMPOUNDS EXHIBITING PROLYL HYDROXYLASE INHIBITORY ACTIVITY, COMPOSITIONS, AND USES THEREOF AMGEN INC. (US) 2008-06-26 WO disclosed