SCHEMBL3830645

SCHEMBL3830645

CC(Br)Oc1ccc2c(c1)C(C)CN(C(=O)C(F)(F)F)CC2

nearest known ligand 0.48

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 4/20 0.48
ESR2 Q92731 4/20 0.48
ABHD6 Q9BV23 4/20 0.40
MTNR1B P49286 10/20 0.37
MTNR1A P48039 8/20 0.37
XIAP P98170 1/20 0.37
BIRC2 Q13490 1/20 0.37
NQO2 P16083 6/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3830648 0.83 ESR1 (0.47) ESR1ESR2ABHD6MTNR1BMTNR1A
SCHEMBL1095205 0.82 ESR1 (0.46) ESR1ESR2ABHD6XIAPBIRC2
SCHEMBL3282323 0.79 ESR1 (0.49) ESR1ESR2
SCHEMBL1095555 0.79 ESR1 (0.49) ESR1ESR2
SCHEMBL3282297 0.79 ESR1 (0.49) ESR1ESR2
SCHEMBL31121204 0.79 ESR1 (0.49) ESR1ESR2
SCHEMBL1095106 0.77 HTR2C (0.51) ESR1ESR2ABHD6MTNR1B
SCHEMBL1095168 0.77 ESR1 (0.52) ESR1ESR2ABHD6XIAPBIRC2
SCHEMBL4937667 0.77 ESR1 (0.65) ESR1ESR2ABHD6MTNR1B
SCHEMBL1095538 0.77 ESR1 (0.65) ESR1ESR2ABHD6MTNR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1833473-B1 5HT2C RECEPTOR MODULATOR COMPOSITIONS AND METHODS OF USE ARENA PHARM INC (US) 2009-09-09 EP disclosed