SCHEMBL3832071

SCHEMBL3832071

C#Cc1ccc(N2CCC(Oc3ccccc3F)C2)nn1

nearest known ligand 0.52

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
SCD O00767 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14130868 1.00 CYP3A4 (0.42) CYP3A4CYP2D6SCD
SCHEMBL5107571 1.00 CYP3A4 (0.42) CYP3A4CYP2D6SCD
SCHEMBL14130994 0.93 CYP3A4 (0.48) CYP3A4CYP2D6
SCHEMBL14130731 0.82 CYP3A4 (0.42) CYP3A4CYP2D6SCD
SCHEMBL3830322 0.82 CYP3A4 (0.42) CYP3A4CYP2D6SCD
SCHEMBL3828538 0.82 CYP3A4 (0.42) CYP3A4CYP2D6SCD
SCHEMBL14130910 0.82 CYP3A4 (0.38) CYP3A4CYP2D6
SCHEMBL3832784 0.82 CYP3A4 (0.38) CYP3A4CYP2D6
SCHEMBL3831365 0.82 CYP3A4 (0.38) CYP3A4CYP2D6
SCHEMBL27784539 0.81 CYP3A4 (0.45) CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2099755-A2 ACETYLENE DERIVATIVES AS STEAROYL COA DESATURASE INHIBITORS Glenmark Pharmaceuticals S.A. (CH) 2009-09-16 EP disclosed
WO-2008062276-A2 ACETYLENE DERIVATIVES AS STEAROYL COA DESATURASE INHIBITORS GLENMARK PHARMACEUTICALS S.A. (US) 2008-05-29 WO disclosed