SCHEMBL3833407

SCHEMBL3833407

CC(C)C(=O)NS(=O)(=O)c1ccc(NC(=O)Cc2ccc(Cl)c(Oc3cc(Cl)cc(C#N)c3)c2F)c(Cl)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.42
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
SLC22A12 Q96S37 1/20 0.36
CA1 P00915 6/20 0.36
CA2 P00918 6/20 0.36
CA12 O43570 4/20 0.36
CA9 Q16790 4/20 0.36
RORC P51449 3/20 0.36
LMNA P02545 1/20 0.34
AKR1C3 P42330 1/20 0.34
AKR1C2 P52895 1/20 0.34
PDK1 Q15118 2/20 0.33
PDK2 Q15119 2/20 0.33
PDK3 Q15120 2/20 0.33
PDK4 Q16654 2/20 0.33
CA5A P35218 1/20 0.33
CA7 P43166 1/20 0.33
CA5B Q9Y2D0 1/20 0.33
MEN1 O00255 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3833330 0.94 CYP3A4 (0.42) CYP3A4CYP2C9CYP2C19SLC22A12RORC
SCHEMBL2637922 0.94 CYP3A4 (0.40) CYP3A4CYP2C9CYP2C19SLC22A12CA1
SCHEMBL2640997 0.94 CYP3A4 (0.40) CYP3A4CYP2C9CYP2C19SLC22A12CA1
SCHEMBL2638552 0.93 CYP3A4 (0.42) CYP3A4CYP2C9CYP2C19SLC22A12CA1
SCHEMBL2639248 0.92 CYP3A4 (0.46) CYP3A4CYP2C9CYP2C19SLC22A12CA1
SCHEMBL2638424 0.92 CYP3A4 (0.43) CYP3A4CYP2C9CYP2C19SLC22A12CA1
SCHEMBL5169997 0.92 CYP3A4 (0.39) CYP3A4CYP2C9CYP2C19SLC22A12CA1
SCHEMBL5170005 0.92 CYP3A4 (0.39) CYP3A4CYP2C9CYP2C19SLC22A12CA1
SCHEMBL2638373 0.91 CYP3A4 (0.41) CYP3A4CYP2C9CYP2C19SLC22A12CA1
SCHEMBL2639193 0.91 CYP3A4 (0.42) CYP3A4CYP2C9CYP2C19SLC22A12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1742908-B1 NON-NUCLEOSIDE REVERSE TRANSCRIPTASE INHIBITORS HOFFMANN LA ROCHE (CH) 2009-11-11 EP claimed