SCHEMBL3834535

SCHEMBL3834535

OC[C@H]1CCCN1c1cc(N2CCc3c(-c4cccc(O)c4)nc(N4CCOCC4)nc32)ccn1

nearest known ligand 0.67

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 20/20 0.67
PIK3R1 P27986 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3834555 1.00 PIK3CA (0.67) PIK3CAPIK3R1
Trifluoroacetic Acid SCHEMBL2377705 0.94 PIK3CA (0.60) PIK3CA
SCHEMBL2377316 0.86 PIK3CA (0.82) PIK3CAPIK3R1
SCHEMBL2377709 0.86 PIK3CA (0.51) PIK3CA
SCHEMBL2378420 0.85 PIK3CA (0.69) PIK3CAPIK3R1
SCHEMBL2375993 0.84 PIK3CA (0.73) PIK3CA
SCHEMBL3831151 0.84 PIK3CA (0.78) PIK3CAPIK3R1
SCHEMBL12247634 0.83 PIK3CA (0.69) PIK3CA
SCHEMBL2378966 0.83 PIK3CA (0.71) PIK3CA
SCHEMBL12247649 0.83 PIK3CA (0.78) PIK3CAPIK3R1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2050749-B1 PYRIMIDINE DERIVATIVE AS PI3K INHIBITOR AND USE THEREOF CHUGAI PHARMACEUTICAL CO LTD (JP) 2017-11-22 EP claimed
EP-2050749-A1 PYRIMIDINE DERIVATIVE AS PI3K INHIBITOR AND USE THEREOF CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2009-04-22 EP claimed