SCHEMBL3835549

SCHEMBL3835549

CCOC(=O)ON1CCC(Nc2ccc(C(=O)c3cc(F)c(Cl)cc3OC)c(N)n2)CC1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 17/20 0.45
CDK4 P11802 16/20 0.45
CCND1 P24385 16/20 0.45
CDK2 P24941 16/20 0.45
MAP4K4 O95819 1/20 0.40
NOS1 P29475 2/20 0.38
NOS2 P35228 2/20 0.38
NOS3 P29474 1/20 0.37
CASK O14936 1/20 0.37
ROCK2 O75116 1/20 0.37
CDKL5 O76039 1/20 0.37
STK10 O94804 1/20 0.37
CDK14 O94921 1/20 0.37
ABL1 P00519 1/20 0.37
EGFR P00533 1/20 0.37
MAK P20794 1/20 0.37
CDK11B P21127 1/20 0.37
TTK P33981 1/20 0.37
CLK1 P49759 1/20 0.37
CLK2 P49760 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3839647 0.92 CDK1 (0.46) CDK1CDK4CCND1CDK2MAP4K4
SCHEMBL3840651 0.90 CDK1 (0.56) CDK1CDK4CCND1CDK2MAP4K4
SCHEMBL3839197 0.88 CDK1 (0.53) CDK1CDK4CCND1CDK2MAP4K4
SCHEMBL3839706 0.85 CDK1 (0.54) CDK1CDK4CCND1CDK2CASK
SCHEMBL3837839 0.85 CDK1 (0.49) CDK1CDK4CCND1CDK2MAP4K4
SCHEMBL3839661 0.85 CDK1 (0.59) CDK1CDK4CCND1CDK2MAP4K4
SCHEMBL3839722 0.84 CDK1 (0.54) CDK1CDK4CCND1CDK2MAP4K4
SCHEMBL3835722 0.84 CDK1 (0.64) CDK1CDK4CCND1CDK2CASK
SCHEMBL3840384 0.82 CDK1 (0.55) CDK1CDK4CCND1CDK2MAP4K4
SCHEMBL3837821 0.82 CDK1 (0.52) CDK1CDK4CCND1CDK2MAP4K4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1771420-B1 NOVEL 2,6-DIAMINOPYRIDINE-3-ONE DERIVATIVES HOFFMANN LA ROCHE (CH) 2009-10-14 EP claimed