SCHEMBL3835798

SCHEMBL3835798

CNC(=O)C=C1C=CC=C(Nc2ncc(F)c(Nc3cccc(-c4nnn[nH]4)c3)n2)C1=O

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
EGFR P00533 15/20 0.42
ITK Q08881 12/20 0.42
BTK Q06187 3/20 0.41
SYK P43405 3/20 0.40
AURKA O14965 1/20 0.38
JAK3 P52333 2/20 0.38
JAK2 O60674 1/20 0.38
LYN P07948 1/20 0.38
TEC P42680 1/20 0.38
TXK P42681 1/20 0.38
BMX P51813 1/20 0.38
CD69 Q07108 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL656118 0.84 EGFR (0.47) EGFRITKBTKSYKAURKA
SCHEMBL656581 0.83 EGFR (0.49) EGFRITKBTKSYKAURKA
SCHEMBL3838652 0.82 SYK (0.49) EGFRITKBTKSYK
SCHEMBL657968 0.81 EGFR (0.50) EGFRITKBTKSYKAURKA
SCHEMBL656244 0.81 EGFR (0.45) EGFRITKBTKSYKAURKA
SCHEMBL3834043 0.80 EGFR (0.62) EGFRITKBTKSYK
SCHEMBL657554 0.77 SYK (0.50) EGFRITKSYKAURKA
SCHEMBL656773 0.75 SYK (0.69) SYKAURKA
SCHEMBL656709 0.75 EGFR (0.44) EGFRITKBTKSYKAURKA
SCHEMBL657135 0.75 SYK (0.53) EGFRITKBTKSYKAURKA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2130541-A2 Methods of treating or preventing autoimmune diseases with 2,4-pyrimidinediamine compounds Rigel Pharmaceuticals, Inc. (US) 2009-12-09 EP claimed