SCHEMBL3836049

SCHEMBL3836049

CCNC(=O)ON1CCC(Nc2ccc(C(=O)c3ccccc3F)c(N)n2)CC1

nearest known ligand 0.52

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 15/20 0.52
CDK4 P11802 14/20 0.52
CCND1 P24385 14/20 0.52
CDK2 P24941 14/20 0.52
MAP4K4 O95819 1/20 0.38
OPRK1 P41145 1/20 0.36
NOS2 P35228 1/20 0.36
ALDH1A1 P00352 1/20 0.36
OPRM1 P35372 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3841223 0.90 CDK1 (0.50) CDK1CDK4CCND1CDK2MAP4K4
SCHEMBL3839661 0.88 CDK1 (0.59) CDK1CDK4CCND1CDK2MAP4K4
SCHEMBL3841254 0.86 CDK2 (0.57) CDK1CDK4CCND1CDK2MAP4K4
SCHEMBL3836160 0.84 CDK1 (0.53) CDK1CDK4CCND1CDK2MAP4K4
SCHEMBL3841297 0.83 CDK1 (0.74) CDK1CDK4CCND1CDK2MAP4K4
SCHEMBL3835552 0.82 CDK1 (0.58) CDK1CDK4CCND1CDK2MAP4K4
SCHEMBL3837689 0.82 CDK2 (0.56) CDK1CDK4CCND1CDK2
SCHEMBL3836156 0.81 CDK1 (0.56) CDK1CDK4CCND1CDK2MAP4K4
SCHEMBL3842619 0.80 CDK1 (0.55) CDK1CDK4CCND1CDK2MAP4K4
SCHEMBL3834933 0.79 CDK1 (0.54) CDK1CDK4CCND1CDK2MAP4K4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1771420-B1 NOVEL 2,6-DIAMINOPYRIDINE-3-ONE DERIVATIVES HOFFMANN LA ROCHE (CH) 2009-10-14 EP claimed