SCHEMBL3841035

SCHEMBL3841035

O=C([C@@H]1C[C@H](N2CCN(c3ccc([N+](=O)[O-])cn3)CC2)CN1)N1CCC(F)(F)C1

nearest known ligand 0.73

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 20/20 0.73
DPP8 Q6V1X1 12/20 0.73
DPP7 Q9UHL4 10/20 0.73
DPP9 Q86TI2 3/20 0.64
FAP Q12884 1/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3847095 0.85 DPP4 (0.78) DPP4DPP8DPP7DPP9FAP
Hydrochloric Acid SCHEMBL2710259 0.85 DPP4 (0.77) DPP4DPP8DPP7DPP9
SCHEMBL3841337 0.85 DPP4 (1.00) DPP4DPP8DPP7DPP9FAP
SCHEMBL3844868 0.83 DPP4 (0.75) DPP4DPP8DPP7DPP9FAP
SCHEMBL3849234 0.83 DPP4 (0.79) DPP4DPP8DPP7DPP9FAP
SCHEMBL3842842 0.82 DPP4 (0.93) DPP4DPP8DPP7DPP9FAP
Hydrochloric Acid SCHEMBL2709769 0.81 DPP4 (0.98) DPP4DPP8DPP9
SCHEMBL3846398 0.80 DPP4 (1.00) DPP4DPP8DPP7DPP9FAP
SCHEMBL3842814 0.79 DPP4 (0.72) DPP4DPP8DPP7DPP9FAP
SCHEMBL3861833 0.79 DPP4 (0.69) DPP4DPP8DPP7DPP9FAP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 27 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10792853-B2 Method and device for producing a 3-D substrate coated with a laminate LEONHARD KURZ STIFTUNG & CO. KG (DE) 2020-10-06 US claimed
US-20200276747-A9 METHOD AND DEVICE FOR PRODUCING A 3-D SUBSTRATE COATED WITH A LAMINATE LEONHARD KURZ STIFTUNG & CO. KG (DE) 2020-09-03 US claimed
US-20180207853-A1 METHOD AND DEVICE FOR PRODUCING A 3-D SUBSTRATE COATED WITH A LAMINATE NIEBLING CURT (DE) 2018-07-26 US claimed
EP-2131830-B1 PHARMACEUTICAL FORM WITH IMPEDED ABUSE GRUENENTHAL GMBH (DE) 2017-05-10 EP claimed
EP-2131830-A2 PHARMACEUTICAL FORM WITH IMPEDED ABUSE Grünenthal GmbH (DE) 2009-12-16 EP claimed
WO-2008107149-A2 PHARMACEUTICAL FORM WITH IMPEDED ABUSE Grünenthal GmbH (DE) 2008-09-12 WO claimed
US-11351718-B2 Overmoulding by 3D printing PLASTIC OMNIUM ADVANCED INNOVATION AND RESEARCH (BE) 2022-06-07 US disclosed
US-20190283314-A1 OVERMOULDING BY 3D PRINTING PLASTIC OMNIUM ADVANCED INNOVATION AND RESEARCH (BE) 2019-09-19 US disclosed
EP-2131830-B1 PHARMACEUTICAL FORM WITH IMPEDED ABUSE GRUENENTHAL GMBH (DE) 2017-05-10 EP disclosed
EP-2116541-B1 Proline derivatives and their use as dipeptidyl peptidase IV inhibitors PFIZER PROD INC (US) 2015-02-25 EP disclosed
EP-1786403-B1 ORAL DOSAGE FORM SAFEGUARDED AGAINST ABUSE CONTAINING (1R, 2R)-3-(3-DIMETHYLAMINO-1-ETHYL-2-METHYL-PROPYL)-PHENOL GRUENENTHAL GMBH (DE) 2013-07-24 EP disclosed
EP-1765303-B1 ORAL DOSAGE FORM SAFEGUARDED AGAINST ABUSE GRUENENTHAL GMBH (DE) 2013-02-20 EP disclosed
EP-1765298-B1 METHOD FOR PRODUCING A SOLID DOSAGE FORM, WHICH IS SAFEGUARDED AGAINST ABUSE, WHILE USING A PLANETARY GEAR EXTRUDER GRUENENTHAL GMBH (DE) 2012-10-24 EP disclosed
EP-1699440-A1 METHOD FOR THE PRODUCTION OF AN ADMINISTRATION FORM WHICH IS SECURED AGAINST MISUSE Grünenthal GmbH (DE) 2006-09-13 EP disclosed
WO-2006002883-A1 METHOD FOR PRODUCING A SOLID DOSAGE FORM, WHICH IS SAFEGUARDED AGAINST ABUSE, WHILE USING A PLANETARY GEAR EXTRUDER Grünenthal GmbH (DE) 2006-01-12 WO disclosed
WO-2006002886-A1 ORAL DOSAGE FORM SAFEGUARDED AGAINST ABUSE CONTAINING (1R, 2R)-3-(3-DIMETHYLAMINO-1-ETHYL-2-METHYL-PROPYL)-PHENOL Grünenthal GmbH (DE) 2006-01-12 WO disclosed
WO-2006002884-A1 ORAL DOSAGE FORM SAFEGUARDED AGAINST ABUSE Grünenthal GmbH (DE) 2006-01-12 WO disclosed
WO-2005063214-A1 METHOD FOR THE PRODUCTION OF AN ADMINISTRATION FORM WHICH IS SECURED AGAINST MISUSE Grünenthal GmbH (DE) 2005-07-14 WO disclosed
EP-0639631-B1 Process for preparing syngas CELANESE GMBH (DE) 1999-11-24 EP disclosed
EP-0639631-A1 Process for preparing syngas HOECHST AKTIENGESELLSCHAFT (DE) 1995-02-22 EP disclosed