SCHEMBL3841871

SCHEMBL3841871

CC(C)(C)C(c1cc2c(cn1)OCCO2)N(C(=O)O)C1CCN(CCn2c(=O)sc3ccc(Cl)cc32)CC1

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TMEM97 Q5BJF2 3/20 0.44
KCNH2 Q12809 4/20 0.38
CYP3A4 P08684 2/20 0.37
CYP2D6 P10635 2/20 0.37
OPRK1 P41145 2/20 0.37
UTS2R Q9UKP6 2/20 0.37
SIGMAR1 Q99720 1/20 0.36
NPY5R Q15761 8/20 0.36
DRD2 P14416 1/20 0.34
DRD4 P21917 1/20 0.34
TACR1 P25103 1/20 0.34
OPRM1 P35372 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4299494 0.81 TMEM97 (0.48) TMEM97KCNH2CYP3A4CYP2D6OPRK1
SCHEMBL3840641 0.76 KCNH2 (0.51) KCNH2
SCHEMBL4294752 0.75 KCNH2 (0.57) TMEM97KCNH2
Hydrochloric Acid SCHEMBL3858458 0.74 KCNH2 (0.56) TMEM97KCNH2
SCHEMBL3840342 0.69 KCNH2 (0.41) KCNH2
SCHEMBL2799505 0.69 KCNH2 (0.34) KCNH2TACR1OPRM1
SCHEMBL3328622 0.69 TSHR (0.34) CYP3A4TACR1
SCHEMBL3149833 0.68 KCNH2 (0.43) KCNH2
SCHEMBL3621094 0.67 KCNH2 (0.44) KCNH2CYP2D6
SCHEMBL3215289 0.67 KCNH2 (0.38) KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2044077-A1 DERIVATIVES AND ANALOGS OF N-ETHYLQUINOLONES AND N-ETHYLAZAQUINOLONES Glaxo Group Limited (GB) 2009-04-08 EP disclosed
WO-2008009700-A1 DERIVATIVES AND ANALOGS OF N-ETHYLQUINOLONES AND N-ETHYLAZAQUINOLONES GLAXO GROUP LIMITED (GB) 2008-01-24 WO disclosed