SCHEMBL3843580

SCHEMBL3843580

Cc1cccc(-c2cnc(O[C@H]3CN4CCC3CC4)nc2)c1

nearest known ligand 0.51

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CHRNA7 P36544 2/20 0.51
ALDH1A1 P00352 1/20 0.48
HTR3A P46098 1/20 0.42
CYP1A2 P05177 1/20 0.40
CYP2D6 P10635 1/20 0.40
CHRM1 P11229 2/20 0.39
CHRM2 P08172 1/20 0.39
CHRM3 P20309 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3843584 1.00 CHRNA7 (0.51) CHRNA7ALDH1A1HTR3ACYP1A2CYP2D6
SCHEMBL16642063 0.91 CHRNA7 (0.44) CHRNA7ALDH1A1HTR3ACHRM1CHRM2
SCHEMBL3844172 0.86 CHRNA7 (0.48) CHRNA7CHRM1CHRM2CHRM3
SCHEMBL3844170 0.86 CHRNA7 (0.48) CHRNA7CHRM1CHRM2CHRM3
SCHEMBL999385 0.86 CHRNA7 (0.64) CHRNA7ALDH1A1CYP1A2CYP2D6CHRM1
SCHEMBL999386 0.86 CHRNA7 (0.64) CHRNA7ALDH1A1CYP1A2CYP2D6CHRM1
SCHEMBL1459611 0.85 CHRNA7 (0.51) CHRNA7CHRM1CHRM2CHRM3
SCHEMBL5397013 0.85 MAP4K4 (0.47) CHRNA7CHRM1CHRM2CHRM3
SCHEMBL3840502 0.85 TSHR (0.49) CHRNA7CHRM1CHRM2CHRM3
SCHEMBL5394680 0.85 MAP4K4 (0.47) CHRNA7CHRM1CHRM2CHRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1537104-B1 AZA-BICYCLOALKYL ETHERS AND THEIR USE AS ALPHA7-NACHR AGONISTS NOVARTIS AG (CH) 2009-11-11 EP claimed
US-9012451-B2 Aza-bicycloalkyl ethers and their use as ALPHA7-nachr agonists NOVARTIS AG (CH) 2015-04-21 US disclosed
US-9012451-B2 Aza-bicycloalkyl ethers and their use as ALPHA7-nachr agonists NOVARTIS AG (CH) 2015-04-21 US disclosed