SCHEMBL3846881

SCHEMBL3846881

C=CCn1c(C)c(C)c2ccnc(NCc3ccc(F)cc3)c21

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 3/20 0.40
CYP2D6 P10635 3/20 0.40
CYP2C19 P33261 3/20 0.40
CYP2C9 P11712 2/20 0.40
CYP3A4 P08684 2/20 0.40
TP53 P04637 2/20 0.38
USP10 Q14694 1/20 0.37
PIK3C3 Q8NEB9 1/20 0.37
USP13 Q92995 1/20 0.37
TDP1 Q9NUW8 2/20 0.36
KDM4E B2RXH2 2/20 0.36
ALDH1A1 P00352 2/20 0.36
HTT P42858 2/20 0.36
MAPT P10636 2/20 0.36
MEN1 O00255 1/20 0.36
GAA P10253 1/20 0.36
HPGD P15428 1/20 0.36
ALOX12 P18054 1/20 0.36
GFER P55789 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL3192695 0.99 CYP1A2 (0.40) CYP1A2CYP2D6CYP2C19CYP2C9CYP3A4
SCHEMBL3838929 0.91 CYP1A2 (0.41) CYP1A2CYP2D6CYP2C19CYP2C9CYP3A4
Hydrochloric Acid SCHEMBL1736575 0.90 CYP1A2 (0.41) CYP1A2CYP2D6CYP2C19CYP2C9CYP3A4
SCHEMBL3844384 0.89 LRRK2 (0.44) CYP1A2CYP2D6CYP2C19CYP2C9CYP3A4
SCHEMBL3843518 0.89 CYP1A2 (0.47) CYP1A2CYP2D6CYP2C19CYP2C9CYP3A4
Hydrochloric Acid SCHEMBL1736394 0.88 LRRK2 (0.43) CYP1A2CYP2D6CYP2C19CYP2C9CYP3A4
Hydrochloric Acid SCHEMBL1736574 0.88 CYP1A2 (0.46) CYP1A2CYP2D6CYP2C19CYP2C9CYP3A4
SCHEMBL3846136 0.87 CYP1A2 (0.44) CYP1A2CYP2D6CYP2C19CYP2C9CYP3A4
Hydrochloric Acid SCHEMBL1737400 0.86 CYP1A2 (0.43) CYP1A2CYP2D6CYP2C19CYP2C9CYP3A4
SCHEMBL3841998 0.86 MAPT (0.44) CYP1A2CYP2D6CYP2C19CYP2C9CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1784404-A4 PYRROLO[2,3-C]PYRIDINE DERIVATIVES AND PROCESSES FOR THE PREPARATION THEREOF YUHAN CORP (KR) 2009-09-09 EP claimed
JP-2008511621-A 2008-04-17 JP claimed
EP-1784404-A1 PYRROLO[2,3-C]PYRIDINE DERIVATIVES AND PROCESSES FOR THE PREPARATION THEREOF Yuhan Corporation (KR) 2007-05-16 EP claimed
WO-2006025716-A1 PYRROLO[2,3-C]PYRIDINE DERIVATIVES AND PROCESSES FOR THE PREPARATION THEREOF YUHAN CORPORATION (KR) 2006-03-09 WO claimed