SCHEMBL3848165

SCHEMBL3848165

COC(=O)OC1(O)CCN(Cc2ccccc2)CC1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 8/20 0.54
ALDH1A1 P00352 3/20 0.54
OPRL1 P41146 1/20 0.52
CYP3A4 P08684 4/20 0.51
POLB P06746 2/20 0.51
HSD17B10 Q99714 1/20 0.51
CYP2C9 P11712 2/20 0.51
CYP2C19 P33261 2/20 0.51
TSHR P16473 1/20 0.50
MEN1 O00255 2/20 0.49
KMT2A Q03164 2/20 0.49
L3MBTL1 Q9Y468 2/20 0.49
USP2 O75604 1/20 0.49
MAPK1 P28482 1/20 0.49
CHRM2 P08172 2/20 0.49
CHRM3 P20309 2/20 0.49
HDAC4 P56524 1/20 0.49
KCNH2 Q12809 1/20 0.49
HDAC1 Q13547 1/20 0.49
OPRM1 P35372 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27733497 0.86 CYP2D6 (0.53) CYP2D6ALDH1A1OPRL1CYP3A4POLB
SCHEMBL6783745 0.84 CYP2D6 (0.58) CYP2D6ALDH1A1OPRL1CYP3A4POLB
SCHEMBL3849168 0.84 CYP2D6 (0.59) CYP2D6ALDH1A1CYP3A4POLBHSD17B10
SCHEMBL4032706 0.81 TSHR (0.57) CYP2D6ALDH1A1OPRL1CYP3A4CYP2C9
SCHEMBL3498095 0.80 CYP2D6 (0.56) CYP2D6ALDH1A1OPRL1CYP3A4POLB
SCHEMBL15387552 0.79 BCHE (0.66) CYP2D6ALDH1A1OPRM1OPRD1
SCHEMBL2694056 0.78 CYP2D6 (0.54) CYP2D6ALDH1A1OPRL1CYP3A4POLB
SCHEMBL21287577 0.78 KMT2A (0.57) CYP2D6ALDH1A1CYP3A4POLBCYP2C9
SCHEMBL14081425 0.77 CYP2D6 (0.56) CYP2D6ALDH1A1OPRL1CYP3A4POLB
SCHEMBL15320057 0.77 OPRL1 (0.51) CYP2D6ALDH1A1OPRL1CYP3A4POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2054053-A1 BIPHENYL SUBSTITUTED SPIROTETRONIC ACIDS AND THEIR USE FOR THE TREATMENT OF RETROVIRAL DISORDERS AiCuris GmbH & Co. KG (DE) 2009-05-06 EP disclosed
WO-2008022725-A1 BIPHENYL SUBSTITUTED SPIROTETRONIC ACIDS AND THEIR USE FOR THE TREATMENT OF RETROVIRAL DISORDERS AICURIS GMBH & CO. KG (DE) 2008-02-28 WO disclosed