SCHEMBL3853029

SCHEMBL3853029

OC1(c2ccc(Cl)cc2)CCN(c2ncnc3ccc(Br)cc23)CC1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 5/20 0.56
ALDH1A1 P00352 3/20 0.53
NPSR1 Q6W5P4 2/20 0.53
CCR5 P51681 1/20 0.46
LMNA P02545 3/20 0.45
KDM4E B2RXH2 2/20 0.45
L3MBTL1 Q9Y468 2/20 0.45
MEN1 O00255 1/20 0.45
GLA P06280 1/20 0.45
KMT2A Q03164 1/20 0.45
AKT2 P31751 2/20 0.44
GSK3B P49841 2/20 0.44
PDGFRB P09619 1/20 0.43
AKT1 P31749 2/20 0.41
CNR1 P21554 1/20 0.41
CNR2 P34972 1/20 0.41
HPGD P15428 2/20 0.41
POLB P06746 1/20 0.41
MAPT P10636 1/20 0.41
CYP1A2 P05177 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL3851636 0.79 AKT1 (0.58) HTTALDH1A1LMNAKDM4EMEN1
SCHEMBL13874436 0.78 CYP3A4 (0.43) HTTALDH1A1LMNAKDM4EMEN1
SCHEMBL29472072 0.76 HTT (0.76) HTTALDH1A1NPSR1LMNAL3MBTL1
SCHEMBL22715242 0.76 HTT (0.76) HTTALDH1A1NPSR1LMNAL3MBTL1
SCHEMBL30333781 0.75 HTT (0.70) HTTALDH1A1NPSR1LMNAKDM4E
SCHEMBL3115181 0.75 HTT (0.74) HTTALDH1A1NPSR1LMNAL3MBTL1
SCHEMBL3849306 0.74 AKT1 (0.43) HTTALDH1A1LMNAKDM4EMEN1
SCHEMBL30902257 0.73 HTT (0.63) HTTALDH1A1NPSR1LMNAKDM4E
SCHEMBL3846177 0.73 HTT (0.63) HTTALDH1A1NPSR1LMNAKDM4E
SCHEMBL3117120 0.72 HTT (0.70) HTTALDH1A1NPSR1LMNAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2048142-A2 Nitrogen-containing condensed cyclic compound having a pyrazolyl group as a substituent group and pharmaceutical composition thereof Eisai R&D Management Co., Ltd. (JP) 2009-04-15 EP disclosed
EP-1382603-B1 NITROGENOUS FUSED-RING COMPOUND HAVING PYRAZOLYL GROUP AS SUBSTITUENT AND MEDICINAL COMPOSITION THEREOF EISAI R&D MAN CO LTD (JP) 2008-07-23 EP disclosed
US-7074801-B1 Nitrogen-containing condensed cyclic compound having a pyrazolyl group as a substituent group and pharmaceutical composition thereof EISAI CO., LTD. (JP) 2006-07-11 US disclosed
EP-1382603-A1 NITROGENOUS FUSED−RING COMPOUND HAVING PYRAZOLYL GROUP AS SUBSTITUENT AND MEDICINAL COMPOSITION THEREOF Eisai Co., Ltd. (JP) 2004-01-21 EP disclosed