SCHEMBL3853243

SCHEMBL3853243

O=C(/C=C/c1ccn(S(=O)(=O)c2cccc(-c3ccc(OC(=O)O)cc3)c2)c1)NO

nearest known ligand 0.49

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 18/20 0.49
HDAC6 Q9UBN7 16/20 0.49
HDAC2 Q92769 17/20 0.48
HDAC8 Q9BY41 16/20 0.48
HDAC3 O15379 16/20 0.48
HDAC10 Q969S8 15/20 0.48
HDAC11 Q96DB2 14/20 0.48
HDAC9 Q9UKV0 14/20 0.48
HDAC4 P56524 13/20 0.48
HDAC7 Q8WUI4 13/20 0.48
HDAC5 Q9UQL6 13/20 0.48
ABL1 P00519 1/20 0.45
EGFR P00533 1/20 0.45
ERBB2 P04626 1/20 0.45
INSR P06213 1/20 0.45
PDGFRB P09619 1/20 0.45
KDM1A O60341 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3850621 0.91 HDAC1 (0.53) HDAC1HDAC6HDAC2HDAC8HDAC3
SCHEMBL3848328 0.91 HDAC1 (0.59) HDAC1HDAC6HDAC2HDAC8HDAC3
SCHEMBL296547 0.91 HDAC1 (0.55) HDAC1HDAC6HDAC2HDAC8HDAC3
SCHEMBL296548 0.91 HDAC1 (0.55) HDAC1HDAC6HDAC2HDAC8HDAC3
SCHEMBL3145473 0.88 HDAC1 (0.51) HDAC1HDAC6HDAC2HDAC8HDAC3
SCHEMBL3145488 0.88 HDAC1 (0.51) HDAC1HDAC6HDAC2HDAC8HDAC3
SCHEMBL3146007 0.85 HDAC1 (0.58) HDAC1HDAC6HDAC2HDAC8HDAC3
SCHEMBL3146017 0.85 HDAC1 (0.58) HDAC1HDAC6HDAC2HDAC8HDAC3
SCHEMBL296243 0.85 HDAC1 (0.52) HDAC1HDAC6HDAC2HDAC8HDAC3
SCHEMBL296244 0.85 HDAC1 (0.52) HDAC1HDAC6HDAC2HDAC8HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1861365-B1 N-SULPHONYLPYRROLES AND THEIR USE AS HISTONE DEACETYLASE INHIBITORS 4SC AG (DE) 2009-07-01 EP claimed