SCHEMBL3853833

SCHEMBL3853833

CCc1cc(-c2nc(CSc3nc(N)c(C#N)c(C4CCCOC4)c3C#N)cs2)ccc1C(=O)O

nearest known ligand 0.44

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 20/20 0.44
SLC6A3 Q01959 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3845090 1.00 ADORA1 (0.44) ADORA1SLC6A3
SCHEMBL3575738 0.88 ADORA1 (0.49) ADORA1SLC6A3
SCHEMBL3853837 0.84 ADORA1 (0.48) ADORA1SLC6A3
SCHEMBL3572617 0.83 ADORA1 (0.61) ADORA1SLC6A3
SCHEMBL14735654 0.79 ADORA1 (0.37) ADORA1SLC6A3
SCHEMBL13550237 0.79 ADORA1 (0.51) ADORA1SLC6A3
SCHEMBL3842754 0.76 ADORA1 (0.40) ADORA1SLC6A3
SCHEMBL3572722 0.75 ADORA1 (0.50) ADORA1SLC6A3
SCHEMBL13550249 0.73 MEN1 (0.43) ADORA1
SCHEMBL3571933 0.73 ADORA1 (0.65) ADORA1SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2099788-B1 CYCLICALLY SUBSTITUTED 3,5-DICYANO-2-THIOPYRIDINES AND USE THEREOF BAYER IP GMBH (DE) 2013-03-06 EP disclosed
EP-2099788-A1 CYCLICALLY SUBSTITUTED 3,5-DICYANO-2-THIOPYRIDINES AND USE THEREOF Bayer Schering Pharma Aktiengesellschaft (DE) 2009-09-16 EP disclosed
WO-2008064788-A1 CYCLICALLY SUBSTITUTED 3,5-DICYANO-2-THIOPYRIDINES AND USE THEREOF BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2008-06-05 WO disclosed