SCHEMBL3854940

SCHEMBL3854940

CCOc1cc(C(=O)N(C(N)=O)C(=O)c2ccc3c(c2)C(=O)[C@H](C)C2(CCNCC2)O3)cc2c1ccn2OCC

nearest known ligand 0.30

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.30
OPRM1 P35372 1/20 0.30
OPRD1 P41143 1/20 0.30
OPRK1 P41145 1/20 0.30
KCNH2 Q12809 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3857178 0.90 CYP2D6 (0.30) CYP2D6OPRM1OPRD1OPRK1KCNH2
SCHEMBL3854564 0.82 ACACB (0.37) CYP2D6OPRM1OPRD1OPRK1KCNH2
SCHEMBL308346 0.72 HDAC3 (0.43)
SCHEMBL4517085 0.68 ACACB (0.37) CYP2D6OPRM1OPRD1OPRK1KCNH2
SCHEMBL308345 0.65 HDAC3 (0.47)
SCHEMBL309464 0.64 TSHR (0.47)
SCHEMBL3856567 0.63
SCHEMBL309677 0.62 ACACB (0.47)
SCHEMBL4787034 0.62 ACACB (0.39)
SCHEMBL14862297 0.61 PBRM1 (0.42) CYP2D6OPRD1OPRK1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2111406-A1 SUBSTITUTED SPIROCHROMANONE DERIVATIVES AS ACC INHIBITORS Merck & Co., Inc. (US) 2009-10-28 EP claimed
WO-2008088688-A1 SUBSTITUTED SPIROCHROMANONE DERIVATIVES AS ACC INHIBITORS MERCK & CO., INC. (US) 2008-07-24 WO claimed