SCHEMBL3860165

SCHEMBL3860165

CC(C)Oc1cccc(C#CC2CCCCC2)c1

nearest known ligand 0.51

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HAO1 Q9UJM8 7/20 0.51
ACACB O00763 2/20 0.46
KCNH2 Q12809 1/20 0.44
BACE1 P56817 1/20 0.42
PTGES O14684 2/20 0.41
PDGFRB P09619 1/20 0.40
PDGFRA P16234 1/20 0.40
GRM5 P41594 2/20 0.40
CYP1A2 P05177 1/20 0.40
MEN1 O00255 1/20 0.39
GAA P10253 1/20 0.39
HTT P42858 1/20 0.39
KMT2A Q03164 1/20 0.39
FFAR1 O14842 1/20 0.38
FFAR4 Q5NUL3 1/20 0.38
NPC1 O15118 1/20 0.38
HPGD P15428 1/20 0.38
RAB9A P51151 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3860671 0.99 HAO1 (0.50) HAO1ACACBKCNH2BACE1PTGES
SCHEMBL236004 0.85 HAO1 (0.47) HAO1ACACBKCNH2BACE1PTGES
SCHEMBL236010 0.85 HAO1 (0.47) HAO1ACACBKCNH2BACE1PTGES
SCHEMBL237227 0.84 HAO1 (0.46) HAO1ACACBKCNH2BACE1PTGES
SCHEMBL233852 0.75 HAO1 (0.47) HAO1KCNH2BACE1PDGFRBPDGFRA
SCHEMBL237026 0.75 HAO1 (0.47) HAO1KCNH2BACE1PDGFRBPDGFRA
SCHEMBL235488 0.75 HAO1 (0.47) HAO1KCNH2BACE1PDGFRBPDGFRA
SCHEMBL236498 0.73 HAO1 (0.46) HAO1KCNH2PDGFRBPDGFRAGRM5
SCHEMBL23025713 0.72 HAO1 (0.49) HAO1PTGESFFAR1FFAR4
SCHEMBL3862174 0.72 HAO1 (0.43) HAO1ACACBBACE1PTGESGRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2076122-A2 ALKYNYL PHENYL DERIVATIVE COMPOUNDS FOR TREATING OPHTHALMIC DISEASES AND DISORDERS Acucela, Inc. (US) 2009-07-08 EP disclosed
WO-2009005794-A2 ALKYNYL PHENYL DERIVATIVE COMPOUNDS FOR TREATING OPHTHALMIC DISEASES AND DISORDERS ACUCELA, INC. (US) 2009-01-08 WO disclosed