SCHEMBL3865020

SCHEMBL3865020

CC(C)(C)c1ccc(COc2ccc(-c3ccc(OC(F)(F)F)cc3)cc2NC(=O)C(=O)O)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SERPINE1 P05121 2/20 0.49
EPHX2 P34913 1/20 0.47
NR1H4 Q96RI1 1/20 0.47
PPARD Q03181 4/20 0.46
TRPV1 Q8NER1 1/20 0.44
RXRA P19793 2/20 0.43
RXRB P28702 2/20 0.43
NR4A2 P43354 2/20 0.43
PPARG P37231 1/20 0.43
PPARA Q07869 1/20 0.43
CACNA1H O95180 1/20 0.42
CYP2C9 P11712 1/20 0.42
IDO1 P14902 1/20 0.42
XDH P47989 1/20 0.41
RXRG P48443 1/20 0.41
PTGER4 P35408 1/20 0.41
PSEN1 P49768 2/20 0.41
ALOX5 P09917 1/20 0.41
VCP P55072 1/20 0.41
RAB9A P51151 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2540994 0.99 SERPINE1 (0.48) SERPINE1EPHX2NR1H4PPARDTRPV1
SCHEMBL2540995 0.93 EPHX2 (0.46) SERPINE1EPHX2NR1H4PPARDTRPV1
SCHEMBL2533885 0.92 EPHX2 (0.47) SERPINE1EPHX2NR1H4PPARDTRPV1
SCHEMBL2540485 0.91 EPHX2 (0.46) SERPINE1EPHX2NR1H4PPARDTRPV1
SCHEMBL13581072 0.82 EPHX2 (0.50) SERPINE1EPHX2NR1H4PPARDTRPV1
SCHEMBL2534864 0.81 SERPINE1 (0.52) SERPINE1EPHX2NR1H4PPARDTRPV1
SCHEMBL1242210 0.81 EPHX2 (0.45) SERPINE1EPHX2NR1H4PPARDPPARA
SCHEMBL2539640 0.81 PPARD (0.50) SERPINE1EPHX2NR1H4PPARDRXRA
SCHEMBL13580799 0.80 EPHX2 (0.46) SERPINE1EPHX2NR1H4PPARDTRPV1
SCHEMBL2537365 0.80 SERPINE1 (0.48) SERPINE1EPHX2NR1H4PPARDRXRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2080751-A1 CARBOXYLIC ACID DERIVATIVE Institute of Medicinal Molecular Design, Inc. (JP) 2009-07-22 EP disclosed