SCHEMBL38737

SCHEMBL38737

[C]#CCCCCCCCC

nearest known ligand 0.50

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.50
THRB P10828 1/20 0.50
PTPN7 P35236 3/20 0.39
HMGCR P04035 1/20 0.39
DNM1 Q05193 5/20 0.38
ALDH1A1 P00352 2/20 0.38
LMNA P02545 2/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
HSD17B10 Q99714 1/20 0.38
SLC22A1 O15245 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1610232 1.00 TSHR (0.50) TSHRTHRBPTPN7HMGCRDNM1
SCHEMBL1611700 1.00 TSHR (0.50) TSHRTHRBPTPN7HMGCRDNM1
SCHEMBL384472 1.00 TSHR (0.50) TSHRTHRBPTPN7HMGCRDNM1
SCHEMBL1611665 1.00 TSHR (0.50) TSHRTHRBPTPN7HMGCRDNM1
SCHEMBL1612633 1.00 TSHR (0.50) TSHRTHRBPTPN7HMGCRDNM1
SCHEMBL1610253 1.00 TSHR (0.50) TSHRTHRBPTPN7HMGCRDNM1
SCHEMBL1613181 1.00 TSHR (0.50) TSHRTHRBPTPN7HMGCRDNM1
SCHEMBL131107 1.00 TSHR (0.50) TSHRTHRBPTPN7HMGCRDNM1
SCHEMBL22721290 1.00 TSHR (0.50) TSHRTHRBPTPN7HMGCRDNM1
SCHEMBL38699 1.00

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 2840 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240131040-A1 COMPOSITIONS AND METHODS RELATED TO CANNABINOID ANIONS Natural Extraction Systems, LLC (US) 2024-04-25 US claimed
US-20230089351-A1 METHODS RELATED TO BIOACTIVE AGENTS THAT CONVERT FROM ANIONS TO MOLECULES Natural Extraction Systems, LLC (US) 2023-03-23 US claimed
US-20230073802-A1 COMPOSITIONS AND METHODS RELATED TO CANNABINOID ANIONS Natural Extraction Systems, LLC (US) 2023-03-09 US claimed
US-20220387376-A1 Compositions Comprising Cannabinoid Molecules that are Dissolved in Water-Miscible Solvents NATURAL EXTRACTION SYS LLC (US) 2022-12-08 US claimed
US-20220387351-A1 Compositions and Methods Related to Organic Oxides Natural Extraction Systems, LLC 2022-12-08 US claimed
US-20210360947-A1 COMPOSITIONS AND METHODS RELATED TO EXCIPIENTS AND CANNABINOID FORMULATIONS Natural Extraction Systems, LLC 2021-11-25 US claimed
WO-2021158575-A1 COMPOSITIONS RELATED TO BIOACTIVE AGENTS THAT CONVERT FROM ANIONS TO MOLECULES Natural Extraction Systems, LLC (US) 2021-08-12 WO claimed
WO-2021087291-A1 COMPOSITIONS AND METHODS RELATED TO ORGANIC OXIDES Natural Extraction Systems, LLC (US) 2021-05-06 WO claimed
WO-2021041637-A1 COMPOSITIONS COMPRISING CANNABINOID IONS DISSOLVING IN GLYCEROL Natural Extraction Systems, LLC (US) 2021-03-04 WO claimed
CN-105503897-A Asymmetric benzophenanthrene tri-furan/thiophene, derivate thereof and preparation method UNIV EAST CHINA NORMAL 2016-04-20 CN claimed
EP-1812427-A1 OXADIAZOLE KETONE INHIBITORS OF FATTY ACID AMIDE HYDROLASE The Scripps Research Institute (US) 2007-08-01 EP claimed
EP-1351940-B1 SUBSTITUTED QUINOLINES FOR THE TREATMENT OF PROTOZOAN AND RETROVIRUS CO-INFECTIONS INST RECH DEVELOPPEMENT IRD (FR) 2007-07-25 EP claimed
US-20060100212-A1 Oxadiazole ketone inhibitors of fatty acid amide hydrolase THE SCRIPPS RESEARCH INSTITUTE (US) 2006-05-11 US claimed
WO-2006044617-A1 OXADIAZOLE KETONE INHIBITORS OF FATTY ACID AMIDE HYDROLASE THE SCRIPPS RESEARCH INSTITUTE (US) 2006-04-27 WO claimed
US-20050165052-A1 Substituted quinolines for the treatment of protozoa and retrovirus co-infections INSTITUT DE RECHERCHE POUR LE DEVELOPPEMENT (FR) 2005-07-28 US claimed
EP-0918757-A1 8-HYDROCARBYL SUBSTITUTED BENZODIZOCINE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS PROTEIN KINASE C (=PKC) MODULATORS GEORGETOWN UNIVERSITY (US) 1999-06-02 EP claimed
WO-1997043268-A1 8-HYDROCARBYL SUBSTITUTED BENZODIZOCINE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS PROTEIN KINASE C (=PKC) MODULATORS GEORGETOWN UNIVERSITY (US) 1997-11-20 WO claimed
EP-0528044-B1 Process for producing 4-substituted gamma- lactone, and the so produced novel substances. JAPAN TOBACCO INC (JP) 1997-08-13 EP claimed
US-5374744-A Sex pheronome of Japanese beetle, cupreous chafers; oxidation, reduction, cleavage, cyclization, alkynylation, hydrolysis JAPAN TOBACCO INC. (JP) 1994-12-20 US claimed
EP-0528044-A1 PROCESS FOR PRODUCING 4-SUBSTITUTED $g(g)-LACTONE, AND NOVEL SUBSTANCE JAPAN TOBACCO INC. (JP) 1993-02-24 EP claimed