SCHEMBL3879635

SCHEMBL3879635

CC(C)c1cc(-c2cc(N3CCN(c4ncccc4C(F)(F)F)CC3)nc(N3CCCC3C)n2)ccn1

nearest known ligand 0.47

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 6/20 0.47
GALR2 O43603 4/20 0.42
GALR1 P47211 4/20 0.42
HSD11B1 P28845 2/20 0.40
KHK P50053 2/20 0.38
MAP3K12 Q12852 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3878236 0.86 TRPV1 (0.49) TRPV1GALR2GALR1HSD11B1KHK
SCHEMBL3888879 0.86 TRPV1 (0.49) TRPV1GALR2GALR1KHKMAP3K12
SCHEMBL3879868 0.85 TRPV1 (0.50) TRPV1GALR2GALR1HSD11B1KHK
SCHEMBL3889943 0.84 TRPV1 (0.48) TRPV1GALR2GALR1KHKMAP3K12
SCHEMBL3879931 0.84 PIK3R1 (0.46) TRPV1GALR2GALR1MAP3K12
SCHEMBL3879378 0.84 TRPV1 (0.47) TRPV1GALR2GALR1HSD11B1
SCHEMBL3878216 0.82 TRPV1 (0.48) TRPV1GALR2GALR1KHK
SCHEMBL3876175 0.81 TRPV1 (0.48) TRPV1GALR2GALR1HSD11B1KHK
SCHEMBL3884821 0.81 TRPV1 (0.53) TRPV1GALR2GALR1HSD11B1
SCHEMBL3877016 0.80 TRPV1 (0.44) TRPV1GALR2GALR1KHKMAP3K12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7566712-B2 Biaryl piperazinyl-pyridine analogues NEUROGEN CORPORATION (US) 2009-07-28 US disclosed
US-7566712-B2 Biaryl piperazinyl-pyridine analogues NEUROGEN CORPORATION (US) 2009-07-28 US disclosed
US-7566712-B2 Biaryl piperazinyl-pyridine analogues NEUROGEN CORPORATION (US) 2009-07-28 US disclosed