SCHEMBL3879909

SCHEMBL3879909

Cc1cc(-c2cc(N3CCN(c4ncccc4Cl)C[C@H]3C)nc(N3CCC3C)n2)ccc1F

nearest known ligand 0.50

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 13/20 0.50
MALT1 Q9UDY8 2/20 0.36
HSD11B1 P28845 1/20 0.36
GRM5 P41594 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13761545 0.95 TRPV1 (0.49) TRPV1MALT1HSD11B1GRM5
SCHEMBL3883269 0.95 TRPV1 (0.49) TRPV1MALT1HSD11B1GRM5
SCHEMBL13761558 0.95 TRPV1 (0.49) TRPV1MALT1HSD11B1GRM5
SCHEMBL3888352 0.95 TRPV1 (0.49) TRPV1MALT1HSD11B1GRM5
SCHEMBL3878083 0.95 TRPV1 (0.49) TRPV1MALT1HSD11B1GRM5
SCHEMBL3879735 0.95 TRPV1 (0.49) TRPV1MALT1HSD11B1GRM5
SCHEMBL3878492 0.94 TRPV1 (0.48) TRPV1GRM5
SCHEMBL3945837 0.93 TRPV1 (0.49) TRPV1MALT1HSD11B1
SCHEMBL3881042 0.92 TRPV1 (0.50) TRPV1HSD11B1GRM5
SCHEMBL3887140 0.92 TRPV1 (0.50) TRPV1HSD11B1GRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7566712-B2 Biaryl piperazinyl-pyridine analogues NEUROGEN CORPORATION (US) 2009-07-28 US disclosed
US-7566712-B2 Biaryl piperazinyl-pyridine analogues NEUROGEN CORPORATION (US) 2009-07-28 US disclosed
US-7566712-B2 Biaryl piperazinyl-pyridine analogues NEUROGEN CORPORATION (US) 2009-07-28 US disclosed