SCHEMBL3880912

SCHEMBL3880912

CC(C)Oc1c(CN(C)C)cc(-c2cc3cc(CN4CCCCC4)ccc3[nH]2)c2c1CNC2=O

nearest known ligand 0.45

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 17/20 0.45
AURKA O14965 3/20 0.41
KDR P35968 3/20 0.41
CDK7 P50613 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3880913 0.88 CHEK1 (0.45) CHEK1AURKAKDRCDK7
Hydrochloric Acid SCHEMBL3841706 0.88 CHEK1 (0.44) CHEK1AURKAKDRCDK7
Hydrochloric Acid SCHEMBL3881150 0.85 CHEK1 (0.48) CHEK1AURKAKDRCDK7
Hydrochloric Acid SCHEMBL3861919 0.85 CHEK1 (0.42) CHEK1AURKAKDRCDK7
Hydrochloric Acid SCHEMBL3039717 0.80 CHEK1 (0.55) CHEK1AURKAKDRCDK7
Hydrochloric Acid SCHEMBL3043783 0.79 CHEK1 (0.51) CHEK1AURKAKDRCDK7
Hydrochloric Acid SCHEMBL3874594 0.78 CHEK1 (0.49) CHEK1AURKAKDR
Hydrochloric Acid SCHEMBL3046874 0.78 CHEK1 (0.47) CHEK1AURKAKDR
Hydrochloric Acid SCHEMBL3040009 0.78 CHEK1 (0.51) CHEK1AURKAKDRCDK7
Hydrochloric Acid SCHEMBL3047063 0.77 CHEK1 (0.53) CHEK1AURKAKDRCDK7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2108642-A1 JAK INHIBITOR Kyowa Hakko Kirin Co., Ltd. (JP) 2009-10-14 EP disclosed