SCHEMBL3881289

SCHEMBL3881289

CCC(CC)NCc1ccc2[nH]c(-c3cc(CN(C)C)cc4c3C(=O)NC4)cc2c1

nearest known ligand 0.41

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
AURKA O14965 10/20 0.41
KDR P35968 10/20 0.41
CDK1 P06493 1/20 0.41
PARP1 P09874 1/20 0.35
FFAR1 O14842 1/20 0.33
KDM4E B2RXH2 1/20 0.31
MAPT P10636 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
F7 P08709 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL3874891 0.99 AURKA (0.41) AURKAKDRCDK1PARP1FFAR1
Hydrochloric Acid SCHEMBL3836110 0.87 AURKA (0.48) AURKAKDRCDK1PARP1FFAR1
SCHEMBL3877283 0.84 AURKA (0.40) AURKAKDRCDK1PARP1MAPT
Hydrochloric Acid SCHEMBL3874897 0.83 AURKA (0.40) AURKAKDRCDK1PARP1MAPT
SCHEMBL3855996 0.81 KDR (0.42) AURKAKDRCDK1PARP1FFAR1
Hydrochloric Acid SCHEMBL3860986 0.80 KDR (0.41) AURKAKDRCDK1PARP1FFAR1
Hydrochloric Acid SCHEMBL3839621 0.80 KDR (0.46) AURKAKDRCDK1PARP1KDM4E
SCHEMBL3835222 0.80 KDR (0.62) AURKAKDRCDK1PARP1KDM4E
Hydrochloric Acid SCHEMBL3874594 0.79 CHEK1 (0.49) AURKAKDRCDK1PARP1
Hydrochloric Acid SCHEMBL3856617 0.76 AURKA (0.51) AURKAKDRCDK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2108642-A1 JAK INHIBITOR Kyowa Hakko Kirin Co., Ltd. (JP) 2009-10-14 EP disclosed