SCHEMBL3882162

SCHEMBL3882162

CC(C)Oc1ccc2cc(C(=O)Nc3ccc(CN)cc3)c(=O)oc2c1OC(C)C

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.53
TP53 P04637 1/20 0.53
MEN1 O00255 1/20 0.47
POLB P06746 1/20 0.47
KMT2A Q03164 1/20 0.47
PLEC Q15149 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
PLG P00747 7/20 0.47
KLK1 P06870 7/20 0.47
KLK6 Q92876 7/20 0.47
MAOA P21397 2/20 0.47
MAOB P27338 2/20 0.47
CNR2 P34972 3/20 0.46
NPC1 O15118 1/20 0.45
RAB9A P51151 1/20 0.45
KLKB1 P03952 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3878869 0.94 TP53 (0.59) MAPTTP53PLGKLK1KLK6
SCHEMBL3881597 0.87 S1PR1 (0.54) MAPTTP53MEN1POLBKMT2A
SCHEMBL3882408 0.86 TP53 (0.63) MAPTTP53PLGKLK1KLK6
SCHEMBL4524105 0.83 TP53 (0.55) MAPTTP53MAOAMAOBCNR2
SCHEMBL3881005 0.83 TP53 (0.53) MAPTTP53MAOAMAOBCNR2
SCHEMBL3955610 0.83 TP53 (0.55) MAPTTP53MAOAMAOBCNR2
SCHEMBL3993825 0.82 TP53 (0.59) MAPTTP53MAOAMAOBCNR2
SCHEMBL3880551 0.82 MAPT (0.54) MAPTTP53MAOAMAOBCNR2
SCHEMBL3881940 0.82 MAOB (0.65) MAPTTP53MEN1POLBKMT2A
SCHEMBL3882652 0.82 TP53 (0.58) MAPTTP53MEN1KMT2APLG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090318546-A1 Chromen-2-One Derivatives NOVARTIS AG (CH) 2009-12-24 US claimed
EP-2010511-A1 CHROMEN-2-ONE DERIVATIVES Novartis AG (CH) 2009-01-07 EP claimed
WO-2007115820-A1 CHROMEN-2-ONE DERIVATIVES NOVARTIS AG (CH) 2007-10-18 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090318546-A1 Chromen-2-One Derivatives CYP1A2, CYP4B1, CYP1B1 MAPT 3872/4885TP53 487/4885MEN1 759/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.