SCHEMBL3884097

SCHEMBL3884097

CC1CCC(C)N1c1nc(-c2ccc(F)c(Cl)c2)cc(N2CCN(c3ncccc3C(F)(F)F)CC2)n1

nearest known ligand 0.45

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
GALR2 O43603 4/20 0.44
GALR1 P47211 4/20 0.44
HSD11B1 P28845 6/20 0.42
TRPV1 Q8NER1 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3952712 0.92 GALR2 (0.44) GALR2GALR1HSD11B1TRPV1
SCHEMBL3878916 0.91 GALR2 (0.46) GALR2GALR1HSD11B1TRPV1
SCHEMBL3887132 0.90 MALT1 (0.45) TRPV1
SCHEMBL3884190 0.90 GALR2 (0.42) GALR2GALR1HSD11B1TRPV1
SCHEMBL3879378 0.90 TRPV1 (0.47) GALR2GALR1HSD11B1TRPV1
SCHEMBL3880207 0.89 GALR2 (0.51) GALR2GALR1HSD11B1TRPV1
SCHEMBL3884990 0.89 GALR2 (0.44) GALR2GALR1HSD11B1TRPV1
SCHEMBL3876175 0.89 TRPV1 (0.48) GALR2GALR1HSD11B1TRPV1
SCHEMBL3879911 0.88 GALR2 (0.42) GALR2GALR1HSD11B1TRPV1
SCHEMBL3876780 0.87 GALR2 (0.46) GALR2GALR1HSD11B1TRPV1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7566712-B2 Biaryl piperazinyl-pyridine analogues NEUROGEN CORPORATION (US) 2009-07-28 US disclosed
US-7566712-B2 Biaryl piperazinyl-pyridine analogues NEUROGEN CORPORATION (US) 2009-07-28 US disclosed
US-7566712-B2 Biaryl piperazinyl-pyridine analogues NEUROGEN CORPORATION (US) 2009-07-28 US disclosed